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N-(1,1-dioxo-1λ6-thian-4-yl)-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
2-[(3-methylbut-2-en-1-yl)(pyridin-2-ylmethyl)amino]butan-1-ol
6-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoate
4-(cyclohexylmethyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,4-diazepane
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
7-methyl-3-[2-(pyrrolidin-3-yl)benzoyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
5-{1-[(2-methoxyphenyl)methyl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
[(2S)-1-{2-[(4-chlorophenyl)methyl]benzoyl}pyrrolidin-2-yl]methanol
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetamide
N-methyl-2-(methylamino)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyridine-4-carboxamide
{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-[(3,4-dimethoxypyridin-2-yl)methyl]azonan-2-one
2-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-3,5-dimethoxybenzoic acid
3-(2-chloro-5-methylphenyl)-1-ethyl-1-(oxan-4-ylmethyl)urea
(2R,6R)-11-methoxy-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(1R,5R)-6-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-[({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}amino)methyl]pyrrolidin-3-ol
1-(2-{1-[(3-methylthiophen-2-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
[(1-methyl-1H-imidazol-2-yl)methyl](3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amine
2-(2,3-dichloro-4-methylphenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
N-(2-methoxyethyl)-4-methyl-3-{[(prop-2-en-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[(2-methylphenyl)methyl]-2-(4-oxo-1,4-dihydroquinolin-1-yl)-N-(prop-2-en-1-yl)acetamide
methyl 2-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]pyridine-3-carboxylate
1-[3-(1H-imidazol-1-yl)propanoyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
[1-(azepan-1-yl)propan-2-yl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
9-[(2-ethoxyphenyl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
2-(2-hydroxyethyl)-8-{[4-(propan-2-yloxy)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-{[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
N-ethyl-6-[3-(hydroxymethyl)piperidin-1-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
N-[(2R,3R)-1'-(1,3-benzothiazol-2-ylmethyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]azetidin-3-yl}piperidine
4-(hydroxymethyl)-1-(5-methylpyrazine-2-carbonyl)azepan-4-ol
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-5,6-dimethylpyridine-3-carboxamide
8-(2-methyl-1H-pyrrole-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
6-fluoro-2-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-{5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
(1R,3S)-7-(6-chloroquinolin-4-yl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}pyridine
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)naphthalene-1-carboxamide
1-[2-amino-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(thiophen-2-yl)ethane-1,2-dione
8-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-benzyl-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S)-N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-(methylsulfanyl)butanamide
(4aS,7aR)-1-(4-hydroxybenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione