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1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
N-(4-methyl-2-oxo-2H-chromen-7-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
N,N-diethyl-2-({4-[(4-hydroxyphenyl)methyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
N-({1-[(2,6-dimethylphenyl)methyl]piperidin-3-yl}methyl)methanesulfonamide
1-(5-methoxy-2-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-(cyclohexylmethyl)-N-ethyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-ethyl-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
N-{4-[2-(1H-imidazol-4-yl)acetamido]phenyl}-5-methylfuran-3-carboxamide
6-(2-{[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino}ethyl)-2-methyl-3,4-dihydropyrimidin-4-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-imidazole-5-carboxamide
3-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
3-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
N-(1H-imidazol-2-ylmethyl)-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-(4-{1-[2-(1H-imidazol-5-yl)ethyl]-3-phenyl-1H-1,2,4-triazol-5-yl}piperidin-1-yl)ethan-1-one
2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}quinolin-4-ol
2-[2-(1H-imidazol-4-yl)ethyl]-9-(propane-2-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-amino-1-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(1H-imidazol-4-yl)propan-1-one
4-(1-ethyl-1H-pyrazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
7-fluoro-2-oxo-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,2-dihydroquinoline-4-carboxamide
1-cyclohexyl-5-(4-methyl-1,3-thiazol-5-yl)-1H-1,2,4-triazole
(1R,5S)-6-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-6-azabicyclo[3.2.1]octane
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]acetamide
5-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(2-methoxyphenyl)methyl]piperazin-2-one
2-methyl-1-[1-(5-methyl-1,3-oxazole-4-carbonyl)azetidin-3-yl]piperidine
1-(carbamoylmethyl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
3-[2-(3,4-difluorophenyl)ethyl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
1-[(4-methoxyphenyl)methyl]-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
5-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
1-methyl-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-fluoro-6-methyl-2-[4-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
7-(cyclohex-1-en-1-yl)-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-(4-{[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenyl)acetamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
2-[1-(propan-2-yl)-5-[4-(1H-pyrazol-3-yl)phenyl]-1H-1,2,4-triazol-3-yl]acetamide
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)benzamide
1-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
N-ethyl-4-[(2-methylpyridin-3-yl)oxy]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
1-(4-aminopyrimidin-2-yl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
N,N,5-trimethyl-2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
N-[(3S,4R)-1-[(3-fluoro-5-methylphenyl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
N-[1-(4-methanesulfonylphenyl)ethyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
(1S,3R)-N-cyclobutyl-3-[2-(phenylsulfanyl)acetamido]cyclopentane-1-carboxamide
1-{6-[4-(thiophene-2-carbonyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
N-methyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(1,2-oxazol-3-ylmethyl)benzamide
1-(4-methanesulfonylpiperazin-1-yl)-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
2-(2-ethyl-1H-imidazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(3-methoxyphenyl)ethyl]pyrrolidin-2-one
N-benzyl-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide