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1-[3-(difluoromethoxy)phenyl]-3-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)urea
1-[4-(1,4-oxazepane-4-sulfonyl)benzoyl]pyrrolidin-3-amine
N-[3-fluoro-4-(trifluoromethyl)phenyl]-4-(2-propoxyethyl)piperazine-1-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
3-({[(4-cyclohexylphenyl)carbamoyl]amino}methyl)-1,2,4-oxadiazole-5-carboxamide
4-(4-phenyl-1H-pyrazol-5-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
4-{5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]pyrimidin-2-yl}morpholine
9-(2-hydroxy-3-methylbutanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-chloro-2-fluoro-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-1,2-dimethylpiperazine
8-methoxy-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-(1-butyl-4-methyl-1H-pyrazol-5-yl)acetamide
N-[(3R,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
(3R,4R)-3-cyclobutyl-4-methyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-3-ol
2-(4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
4-[1-(2-methoxy-5-methylbenzenesulfonyl)azetidin-3-yl]pyridine
5-(2,2-diphenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(3-methoxyphenoxy)ethan-1-one
4-{3-[4-(1H-imidazol-2-yl)phenoxy]propyl}morpholine
(1S,6R)-N-(2-methoxyphenyl)-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
1-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-4-(piperidin-1-yl)piperidine
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
9-[2-(4-methoxyphenoxy)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-cyclopentyl-N,1-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]propanamide
3-(2-{2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)imidazolidine-2,4-dione
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[4-(methylamino)pyrimidin-2-yl]-decahydro-1,6-naphthyridin-2-one
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]naphthalene-1-carboxamide
N-[2-(dimethylamino)ethyl]-5-hydroxy-N-[(5-methylthiophen-2-yl)methyl]pyrazine-2-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{3-[(2-methylphenyl)methyl]-1,2,4-oxadiazol-5-yl}phenyl)-1,3-diazinane-2,4-dione
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(quinolin-4-yl)pyrrolidin-3-yl]acetamide
3-amino-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
N-(1H-imidazol-2-ylmethyl)-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[5-(4-chlorophenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-{[4-(methylsulfanyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-oxo-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
5-cyclopropanecarbonyl-1'-[(3-fluoro-4-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,5S,8S)-3-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-8-methoxy-3-azabicyclo[3.2.1]octane
(1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(hydroxymethyl)piperidin-3-yl)methanol
2-(pyridin-4-yl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-4-acetamidobutanamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
5-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
N-[2-(3-methoxyphenyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
9-[2-oxo-2-(piperazin-1-yl)ethyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one