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2-(ethylsulfanyl)-5-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyrimidine
4-[(5-methylfuran-2-yl)methyl]-3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
3-(2,3-dimethoxyphenyl)-N,N-diethyl-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
[(2S,6S)-4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
methyl 4-[(4-{2-[(pyridin-3-ylmethyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
N2-benzyl-N2,7,7-trimethyl-N5-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
3-[1-(3-hydroxybenzoyl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-dimethyl-5-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-N-[2-(pyridin-3-yl)ethyl]piperidin-4-amine
3-(5-chloro-4-oxo-3,4-dihydroquinazolin-3-yl)-1λ6-thiolane-1,1-dione
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
3-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[4-(pyrrolidine-1-carbonyl)morpholin-3-yl]acetamide
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-methylphenyl)piperazine
3-[(4-methyl-1,4-diazepan-1-yl)methyl]-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
7-chloro-4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(4-{1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}butan-2-yl)-4-methylpiperazine
methyl 3-({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}sulfamoyl)thiophene-2-carboxylate
3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-5,6-dimethyl-1,2-dihydropyridin-2-one
1-[4-(4-{furo[3,2-c]pyridin-4-yl}piperazin-1-yl)piperidin-1-yl]butan-1-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]pyrazine-2-carboxamide
(2S)-N-[3-(2-methoxyphenyl)propyl]-5-oxopyrrolidine-2-carboxamide
(3R,4R)-3-cyclopropyl-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-methylpyrrolidin-3-ol
(2R)-2-amino-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-methylpentanamide
N-{3-[1-(3-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]propyl}acetamide
N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,3-dihydro-1H-indene-1-carboxamide
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2,4-dimethylpyrimidine-5-carboxamide
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-2-(pyridin-3-yl)ethan-1-one
7-methoxy-3-(1H-pyrazole-4-sulfonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2,2-dimethylthiomorpholin-3-one
4-(1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-3-yl)benzoic acid
2-{4-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-ol
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine
2,5,6-trimethyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}pyrimidin-4-amine
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
2-[(3-chlorophenyl)methyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,3-benzoxazole-6-carboxamide
6-({4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}methyl)-1H-indole
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(naphthalen-1-yl)urea
2,2-dimethyl-5-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)pentan-1-ol
2-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
2-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]-3,4,7-trimethyl-1H-indole
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(piperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-{[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]formamido}ethyl)propanamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methyl-1H-1,3-benzodiazole-5-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2,3,4-tetrahydronaphthalene-2-carboxamide