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({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
2,6-dimethyl-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
5-[1-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
3-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
7-chloro-4-hydroxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]quinoline-3-carboxamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N-ethylpyridine-4-carboxamide
{8-methyl-2-[4-(1-propylpiperidin-4-yl)piperazin-1-yl]quinolin-3-yl}methanol
1-cyclohexyl-N-(2-methylpropyl)-4-oxo-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
5-oxo-1-[2-(pyridin-2-ylmethoxy)phenyl]pyrrolidine-3-carboxylic acid
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-2-(2-{[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]formamido}ethyl)-1,3-thiazole-5-carboxylic acid
1-ethyl-N-(1,4-oxazepan-6-ylmethyl)-1H-pyrazole-4-sulfonamide
5-{[4-(4-fluorophenoxy)piperidin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
1-(cyclohex-3-ene-1-carbonyl)-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-(3-chlorophenyl)-4-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}piperazine
3-{1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]azetidin-3-yl}pyridine
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-[(4-phenyloxan-4-yl)methyl]pyrimidin-2-amine
2-(2,2-dimethyloxan-4-yl)-4-{3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
methyl 3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
9-(5-methyl-1,2-oxazole-3-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1H-indazol-3-yl)-1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
5-{[benzyl(methyl)amino]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
1-{1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
N-[(2-fluorophenyl)methyl]-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}propanamide
3-(2-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-4-(2-methylpropyl)piperazin-2-one
1-methyl-4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-indole
1-(2,3-dihydro-1H-inden-2-yl)-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,4-diazepane
4-methoxy-3-(2-phenoxyethyl)benzamide
N-(pyridin-2-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
9-[2-(2-oxopiperidin-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1H-1,3-benzodiazol-2-ylmethyl)(ethyl)({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]benzonitrile
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(pyridin-4-ylmethyl)urea
5-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-2-methyl-2H-1,2,3,4-tetrazole
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
2-[4-(2,2-dimethylpropyl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
7-(5-methyl-4-phenylthiophene-3-carbonyl)-2-oxa-7-azaspiro[4.5]decane
4-hydroxy-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-({5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}methyl)pyridine
5-(3-cyclopropyl-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)-1H-1,2,4-triazole
2-methyl-2-[4-(morpholin-4-yl)-2-(pyrrolidin-1-yl)pyrimidin-5-yl]propanoic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(methoxymethyl)furan-2-carboxamide
N-{[1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
2-benzyl-9-(pent-4-enoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-fluoro-N-[1-(methoxymethyl)cyclopentyl]quinoline-2-carboxamide