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3-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,4-diazepane
2-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
4-(2-fluorophenoxy)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylic acid
(2-{2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]acetamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-ethyl-N-methylpyrimidin-4-amine
(2H-1,3-benzodioxol-4-ylmethyl)(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
(5-{1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)propanamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[(3-methylpyridin-4-yl)methyl]-1,3-oxazole-4-carboxamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-3-propyl-1H-pyrazole-5-carboxamide
2-(2,3-dihydro-1H-isoindole-2-carbonyl)-3,5,7-trimethyl-1H-indole
2-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4,5,6-trimethyl-3-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-(2-hydroxybenzoyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(1-methyl-1H-pyrazole-5-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
2-{4-[(3-fluorophenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
6-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(propan-2-yl)pyrimidine-4-carboxamide
N-methyl-5-[4-(piperidin-1-yl)butanoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-(3-chlorophenoxy)-N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
2-cyclopentyl-9-(6-ethyl-2-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-{[1-(pyrazin-2-yl)propan-2-yl]amino}quinazoline-6-carboxylic acid
[3-(2-phenylethyl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]methanol
methyl (2S,4R)-4-(dimethylamino)-1-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)pyrrolidine-2-carboxylate
(2R,4R)-4-hydroxy-N-[2-(4-methoxyphenyl)ethyl]-N-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
1-(1H-imidazol-4-ylmethyl)-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
N-{2-[1-(2-chlorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}acetamide
(1R,5R)-3-(4-chloro-2-fluorobenzoyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
benzyl({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
N-(3-hydroxypropyl)-2-methyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydroquinoline-8-carboxamide
2-({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
8-(morpholine-2-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-[(4-fluorophenyl)methyl]-4-(2-methyloxolane-2-carbonyl)piperazin-2-one
3-(morpholine-4-carbonyl)-1-propyl-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[1-(2-methylpyridin-4-yl)-3-propylpiperidin-3-yl]methanol
1,3-dimethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
6-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-N-methylpyridine-2-carboxamide
(3S,9aR)-3-benzyl-8-(2,3-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2-methylphenyl)-4-[2-(pyridin-4-ylsulfanyl)acetyl]piperazin-2-one
2-cyclohexyl-5-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)pyrimidine
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2,6-dimethylpyrimidine-4-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-(propylsulfanyl)ethan-1-one