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(3R)-3-[1-butyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinoline
6-(azepan-1-yl)-N-(oxan-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(azepan-1-yl)-3-[3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]propan-2-ol
N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-amino-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)cyclobutane-1-carboxamide
5-methyl-4-{2-oxo-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1H-pyrazol-3-one
N-(2,4-difluorophenyl)-3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}benzamide
1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
1-(furan-2-ylmethyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-(propan-2-yl)-4-[4-(thiophen-3-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
3-fluoro-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]pyridine-4-carboxamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
(4aS,8aR)-6-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
(4aS,8aR)-6-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]propanamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[2-(pyrazin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
(2S,4S)-4-cyclopentaneamido-N-ethyl-1-(4-methylpyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
2-{4-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-ol
2-fluoro-6-[3-(2-methoxyphenoxy)propyl]benzamide
(3S)-1-{1-methyl-5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(2-methyl-1,4-oxazepan-4-yl)pyridine-3-carboxamide
N-cyclohexyl-3-{[6-(piperidin-4-yl)pyrimidin-4-yl]amino}propanamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
2-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-6-methylpyridin-3-ol
2-(4-methoxy-2,5-dimethylphenyl)-1-[3-(1H-pyrazol-1-yl)propyl]-1H-imidazole
4-{3-cyclopropyl-5-[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
1-(1-{[1-(thian-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}isoquinoline
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
(3R)-3,4,4-trimethyl-1-[4-(morpholine-4-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
4-[6-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)pyrimidin-4-yl]morpholine
3-[2-(3-methoxyphenyl)phenyl]-1-methyl-1-[2-(morpholin-4-yl)propyl]urea
5-fluoro-2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-hydroxy-N-[(5-methylpyrazin-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
9-methoxy-N-methyl-7-oxo-3-(4-phenylbutanoyl)-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-{5-[2-chloro-5-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
N-[3-(methylsulfanyl)propyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-[4-({[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
1-[2-(dimethylamino)ethyl]-5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}piperidin-2-one
1-[4-(4-{[2-(3-fluorophenyl)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
1-(4-fluorophenyl)-4-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}piperazine
1-{[4-(3,4,5-trimethoxyphenoxy)phenyl]methyl}pyrrolidine
{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}[(2-fluorophenyl)methyl]amine
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4,6-dimethylpyrimidine
1-[(2-methoxyphenyl)methyl]-N3-methyl-N5-(3-methylbutyl)-4-oxo-N3-[1-(1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4S)-4-(3-methoxyphenyl)-1-(quinolin-4-ylmethyl)piperidin-3-ol
4-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]benzene-1-sulfonamide