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4-oxo-4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]butane-1-sulfonamide
5-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)-2,1,3-benzoxadiazole
(2-{methyl[(4-phenoxyphenyl)methyl]amino}-1,3-thiazol-4-yl)methanol
N,N-diethyl-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
1-(2-fluoro-4-methoxyphenyl)-2-(4,4,4-trifluorobutyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-[(5-methylpyrazin-2-yl)methyl]-9-(quinolin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
7,8-dimethyl-4-(3-methylpiperidine-1-carbonyl)-2-(2-methylpyrimidin-5-yl)quinoline
4,4,4-trifluoro-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]butanamide
1-[1-(4-hydroxyphenyl)ethyl]-3-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]urea
(3S)-1-[5-(azocane-1-carbonyl)-1-methyl-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
5-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]furan-2-carboxamide
N'1-(2-methoxyethyl)-N'1-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)cyclopropane-1,1-dicarboxamide
6-methyl-5-(5-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[(3,4,5-trimethoxyphenyl)methyl]morpholine-2-carboxamide
1-tert-butyl-4-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}(methyl)amino)methyl]pyrrolidin-2-one
2-{[(3S,4R)-3-cyclopropyl-4-(3-methoxypropanamido)pyrrolidin-1-yl]methyl}benzoic acid
4-[(3-fluorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
9-[(3,5-dichloro-2-methoxyphenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
6-{4-[1-(2-methylpropyl)piperidin-4-yl]piperazin-1-yl}pyrimidine-2,4-diamine
2-methyl-N-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-({2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(cyclohexylmethyl)-4-[5-(methoxymethyl)furan-2-carbonyl]morpholine
2-(1H-imidazol-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)benzamide
2-amino-4-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropan-1-amine
2-(4-fluorophenyl)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidine
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperidine-1-carboxamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propyl)pyrrolidin-2-one
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[(2-methoxyphenyl)methyl]-2-methyl-N-propyl-5-sulfamoylbenzamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
4-(4-fluorophenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]oxane-4-carboxamide
methyl 1-[2-hydroxy-3-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
2-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]benzonitrile
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(methylamino)pyridine-4-carbonyl]-decahydro-1,6-naphthyridin-2-one
1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(thiophen-2-yl)propan-1-one
(3R,4R)-4-amino-1-({3-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)piperidin-3-ol
7-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3-azaspiro[5.5]undecan-9-amine
2-(3-methoxyphenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(4-fluorophenyl)-4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]butane-1,4-dione
2-(2,4-difluorophenyl)-2-[2-(1-propylpiperidin-4-yl)acetamido]acetic acid
N-(furan-2-ylmethyl)-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
dimethyl(2-{4-[4-(2-methylpropyl)benzoyl]morpholin-2-yl}ethyl)amine