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4-(4-methyl-1H-pyrazol-1-yl)-1-(pyridin-4-yl)piperidine-4-carboxylic acid
(1R,5R)-3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{4-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
3-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-2-methoxybutanamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
methyl 1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-methylbutyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)azetidine
2-[4-(2-methyloxane-2-carbonyl)piperazin-1-yl]-1,3-benzothiazole
5-ethyl-4-{4-[(4-methanesulfonylphenyl)methyl]piperazin-1-yl}-2-methylpyrimidine
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
2-[4-(2-fluoro-5-methoxyphenyl)phenyl]-N-methylacetamide
4-(2-chloro-6-methoxyphenyl)-5-methylthieno[2,3-d]pyrimidine
(2S,4S)-4-amino-N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-1-methylpyrrolidine-2-carboxamide
2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(4-methyl-2-oxopentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(4-methoxyphenyl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-(2-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}ethyl)-N-methylmethanesulfonamide
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-[(1S)-1-phenylethyl]propanamide
9-cyclopentanecarbonyl-1-methyl-4-[(4-methylphenyl)methyl]-1,4,9-triazaspiro[5.5]undecane
3-(pyridin-4-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-{1-[(2,2-diphenylcyclopropyl)methyl]azetidin-3-yl}pyridine
2-(dimethylamino)-1-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-2-(4-methylphenyl)ethan-1-one
N-(2-fluorophenyl)-3-{1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}propanamide
2-amino-6-(2,5-dimethylfuran-3-yl)-4-[2-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
5-(2-chlorophenyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]furan-2-carboxamide
2-(4-fluoro-2-methoxyphenyl)-5-(piperidin-1-ylmethyl)pyridine
2-(1-benzothiophen-3-yl)-4-{1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}pyridine
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(pyridazine-3-carbonyl)-1,4-diazepane
N-{[2-(6-oxo-1,6-dihydropyridin-3-yl)phenyl]methyl}propanamide
N-{3-oxo-3-[3-(3-phenylpropanoyl)piperidin-1-yl]propyl}methanesulfonamide
6-butyl-2-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
1-(methoxymethyl)-N-[1-(2-methoxyphenyl)propan-2-yl]-N-methylcyclobutane-1-carboxamide
4-[({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
2-cyclopropyl-8-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
N-[2-(dimethylamino)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1,5-dimethyl-4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
[3-(2-chlorophenyl)propyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
(4-{[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
methyl 5-{[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
(2S,4S)-4-amino-1-{[1-(4-methoxyphenyl)-1H-pyrrol-2-yl]methyl}-N-methylpyrrolidine-2-carboxamide
(4aR,7aS)-1-methanesulfonyl-4-(5-methoxyfuran-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-phenylethane-1,2-dione
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(4-ethylpiperazin-1-yl)acetamide
(3aS,6aS)-1-methyl-5-(4-pentylbenzenesulfonyl)-octahydropyrrolo[3,4-b]pyrrole