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2-methoxy-5-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl](quinolin-3-ylmethyl)amine
1-[2-(1H-indol-3-yl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{4-ethyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-2-yl}morpholine
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-methyl-2-phenyl-4-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2,3,6-trifluorophenyl)methyl]pyrimidin-2-amine
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-6,8-dimethyl-1,2-dihydroquinolin-2-one
(4aS,7aR)-1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]propanamide
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
1-(2-chlorophenyl)-4-[(2S)-2-hydroxy-3-phenylpropanoyl]piperazin-2-one
N,N-dimethyl-5-{[4-(naphthalen-2-yl)piperazin-1-yl]methyl}-1,3-thiazol-2-amine
1-[(3,4-dimethoxyphenyl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
(2S)-3-methyl-2-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)butan-1-ol
(2S,4S)-4-amino-1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-benzyl-1-{2-[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[(1-hydroxycyclohexyl)methyl]-1H-imidazol-2-yl}-N-methylbenzene-1-sulfonamide
2-(1-methyl-4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
4-[(4-methoxypyridin-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-({1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
5-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}pentanoic acid
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[(2-methylpyridin-4-yl)methyl]urea
methyl (1R,3S,3aR,6aS)-3-(2-ethylphenyl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-ethyl-1-[(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]urea
4-[1-(piperidine-1-sulfonyl)piperidin-3-yl]benzoic acid
[(3R,5R)-1-[5-(methoxymethyl)furan-2-carbonyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-methyl-9-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
N-(butan-2-yl)-3-(2-oxoimidazolidin-1-yl)-N-(thiophen-3-ylmethyl)benzamide
5-ethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-3-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
ethyl 1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-(4-{[3-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
(3R,4R)-4-amino-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
3-butyl-1-methyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperazin-2-one
3-(1,2-oxazinan-2-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
[(2S,6S)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-(3,5-difluoropyridine-2-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
3-[2-(dimethylamino)ethyl]-8-[(3-hydroxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-6-(2-methoxyphenyl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
3-(1-methyl-1H-1,2,4-triazol-3-yl)-1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}urea
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1H-pyrazole-3-carbonyl)piperidine
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-5-ethyl-2-methylpyrimidin-4-amine
6-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole