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1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(3-methoxyphenoxymethyl)piperidine
1-[3-(2-phenylacetyl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
(1S,5R)-6-(2-methylbenzenesulfonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(2-oxopiperidin-3-yl)acetamide
N-methyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
{1-[2-(methylamino)pyridine-4-carbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
5-[(dimethylamino)methyl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
1-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(3,4,5-trimethoxyphenyl)ethan-1-one
4-(1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)benzoic acid
3-(4-fluorophenyl)-N-(1-methanesulfonylpiperidin-4-yl)-3-phenylpropanamide
(2S)-2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}-2-phenylacetamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]benzamide
N-(2-methoxyethyl)-1-{1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(thiophen-2-yl)ethan-1-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)pyridine-3-carboxamide
6-ethyl-N,N-dimethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
(3S,9aR)-8-(3-fluoro-4-methylbenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-(methylamino)pyrimidine-5-carbonyl]-1,4-diazepan-6-ol
2-[1-(furan-2-ylmethyl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazin-2-yl]ethan-1-ol
(3R,4R)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-cyclopropyl-4-phenyl-9-(pyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[4-(morpholin-4-yl)butyl]benzamide
1-(2-methoxyacetyl)-N-{2-[(4-methylphenyl)sulfanyl]ethyl}piperidine-3-carboxamide
({[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methyl}sulfamoyl)dimethylamine
3-(2-amino-5-methylpyridin-3-yl)benzoic acid
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
(3S,4R)-1-(3,4-difluorobenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(5-methylpyrazin-2-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
N-[2-(1-benzofuran-2-yl)pyridin-3-yl]-2-methylpropanamide
1-[(5-methylthiophen-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-(4-{imidazo[1,2-a]pyridine-6-carbonyl}piperazine-1-carbonyl)morpholine
3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-1-[3-(morpholin-4-yl)propyl]urea
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-{1-[(2-fluorophenyl)methyl]azepan-4-yl}-5-methoxy-4-oxo-4H-pyran-2-carboxamide
4-{[(2R,5S)-5-[(3,5-difluoro-4-methoxyphenyl)methyl]oxolan-2-yl]methyl}-1,4-oxazepane
1-(3-chloro-2-propoxyphenyl)-3-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-oxo-4-phenylbutanamide
4-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
2-[1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)pyrrolidin-2-yl]pyridine
methyl 4-[5-({4-[hydroxy(pyridin-3-yl)methyl]piperidin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{[(3S,4S)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-hydroxypiperidin-4-yl]methyl}pyrrolidine-1-carboxamide
6-methoxy-1-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-2-carboxamide
N,N-diethyl-1-[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]pyrrolidin-3-amine
1-ethyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-propyl-1H-pyrazole-4-carboxamide
1-{5-[(4-benzylpiperidin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-methyl-1,4-diazepane