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8-[6-(1-hydroxyethyl)pyridin-2-yl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
6-[4-(hydroxymethyl)piperidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[(3R,4R)-1-(1,3-benzothiazol-2-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
2-{2-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methoxyfuran-2-carboxamide
(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-(2-phenoxyethyl)piperidin-3-yl)methanol
3-(2-hydroxyethyl)-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
methyl[(3-methylpyridin-2-yl)methyl][3-(methylsulfanyl)butyl]amine
4-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
N-ethyl-2-[4-(1H-pyrazole-4-carbonyl)piperazin-1-yl]acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[3-(trimethyl-1H-pyrazol-1-yl)propanamido]acetic acid
(1-methyl-1H-imidazol-2-yl)(1-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}piperidin-4-yl)methanol
2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]naphthalen-1-ol
N-cyclopropyl-2-(6-fluoro-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethyl-1,3-oxazole-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]pyrrolidin-3-yl]-2-propoxyacetamide
4-{1-azabicyclo[3.2.1]octan-5-yloxy}-2,3-dihydro-1H-inden-1-one
2-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-(methoxymethyl)-1H-pyrazol-1-yl}-4-(furan-2-yl)pyrimidine
1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-phenylpiperazine
N-(4-{2-[methyl(pyridin-4-ylmethyl)amino]acetamido}phenyl)pentanamide
methyl 3-hydroxy-2-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanoate
(3S,4S)-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
(2S,4R)-4-amino-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-N-methylpyrrolidine-2-carboxamide
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
7-(3-chlorophenyl)-4-[2-(dimethylamino)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[(2S,4S)-4-fluoro-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-2-yl]methyl}-3,3-dimethylbutanamide
1-(3-chlorophenyl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazine
2-[({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
3-(4-hydroxyphenyl)-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-[3-(furan-2-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazole
N-[(5-methylfuran-2-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-(4-fluorophenyl)-4-(1H-pyrazole-3-carbonyl)-1,4-diazepane
2-{[4-(4-chloro-2-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
1-benzyl-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-(3-methoxyphenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-(2-methoxybutanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
3-(furan-2-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
N,2-dimethyl-3-[(pyridin-3-ylmethyl)amino]-N-[1-(pyrimidin-4-yl)ethyl]benzamide
N-(1H-1,3-benzodiazol-5-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
(4aS,7aR)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-4-{[({2-[(quinoxalin-6-yl)amino]-1,3-thiazol-5-yl}methyl)amino]methyl}pyrrolidin-2-one
4-(2-methoxyethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
3-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-acetamido-N-propyl-N-(pyridin-3-ylmethyl)acetamide
N-[(3,4-dimethoxyphenyl)methyl]-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-[(3aS,6aS)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N-[(4-acetylmorpholin-2-yl)methyl]-3-(pyridin-3-yl)propanamide