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1-ethyl-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidin-2-one
5-(2-methylphenyl)-4-[1-(oxolane-3-carbonyl)piperidin-3-yl]-2-(pyridin-4-yl)pyrimidine
6-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-1,2-oxazole-3-carboxamide
(1S,3R)-3-amino-N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-methoxyethyl)cyclopentane-1-carboxamide
2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]propane-1,3-diol
2-methyl-3-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
1-[(3S)-3-(dimethylamino)azepan-1-yl]-3-(pyridin-2-yl)propan-1-one
1-methyl-3-[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
[(3-chloro-4-fluorophenyl)methyl](methyl)[2-(oxan-2-yl)ethyl]amine
2-(2-hydroxyethyl)-9-[(5-propylfuran-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(5-phenyl-1,3,4-thiadiazol-2-yl)-decahydro-1,6-naphthyridin-2-one
2-butyl-8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-methyl-N-{1-[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
4-{2-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
N-(prop-2-en-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
3-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenol
3-[1-(1H-pyrazol-1-yl)ethyl]-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(2-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-2-yl}ethyl)phenol
[(3R,5R)-5-[(dimethylamino)methyl]-1-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]piperidin-3-yl]methanol
1-methyl-2-oxo-8-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-(2-amino-5-chloro-6-methylpyrimidin-4-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[2-(azepan-1-yl)ethyl]-N,1,3-trimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}dimethylamine
1-propyl-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine
2-{1H-pyrrolo[2,3-b]pyridin-4-yl}quinoxaline
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-(4-methylpentyl)morpholine
2-[(4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)methyl]benzonitrile
N-[1-(2-methylpropyl)cyclopropyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[3-({[2-(4-fluorophenyl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,9aR)-3-(4-aminobutyl)-8-(cyclohexylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(1-benzylpiperidin-3-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1,4-dioxan-2-ylmethyl)({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
N-(2-methyl-1-{7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-methoxy-1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
3,3-dimethyl-1-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}urea
4-[4-(1,3,4-oxadiazol-2-yl)phenyl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
7-methoxy-2-(2-methoxyphenyl)-3-(1H-pyrazol-1-ylmethyl)quinoline
9-[(2-aminopyridin-3-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-(propan-2-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
5-(4-hydroxy-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-N'-phenylethanediamide
4-{4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanoyl}-1λ6-thiomorpholine-1,1-dione
3-benzyl-1-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(5-chlorothiophene-2-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
5-cyclopentyl-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
4-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]benzonitrile
(2S,4S)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-acetamido-N-ethylpyrrolidine-2-carboxamide