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3,5-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]furan-2-carboxamide
[(3S,5R)-1-(morpholine-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-(4-fluorophenyl)-1,4-diazepane
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-ethyl-3-methyl-1H-pyrazol-4-amine
2-amino-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N,1-diethyl-5-methyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1H-pyrazole-4-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
8-methyl-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
(2R,6R)-11-methoxy-4-(5-methylthiophene-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(3-ethoxyphenyl)-2-[4-(1-methyl-1H-imidazole-2-carbonyl)morpholin-3-yl]acetamide
N-(1-cyclopentanecarbonylpiperidin-4-yl)-2-(phenylamino)pyrimidine-5-carboxamide
methyl 5-[(2,3-dihydroxypropyl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-ethyl-6-oxopiperidine-3-carboxamide
(1S,6R)-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-benzyl-8-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-fluoro-4-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]quinazoline
ethyl 4-({[1-(2,2-dimethylpropyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)piperidine-1-carboxylate
N-(furan-2-ylmethyl)-9-methoxy-7-oxo-3-(2-phenoxyacetyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
(3S,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
5-{[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{[4-(2,3-dichlorophenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
(2,1,3-benzoxadiazol-4-ylmethyl)(ethyl)({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amine
1-(4-chlorophenyl)-N-{[1-(cyclopent-3-ene-1-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-2-(1H-1,2,3,4-tetrazol-1-yl)pyridine
3-(N-methylmethanesulfonamido)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
4-chloro-5-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}thian-4-amine
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2,4-dimethoxyphenyl)ethyl]acetamide
ethyl 2-[7-(2-methylbenzoyl)-2,7-diazaspiro[4.5]decan-2-yl]acetate
1-(1H-imidazol-2-ylmethyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
1-(6-fluoroquinolin-8-yl)-4-methylphthalazine
4-[2-amino-3-cyano-6-(1H-pyrrol-3-yl)pyridin-4-yl]benzamide
1-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
methyl 4-({4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}methyl)benzoate
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-3-propyl-1H-pyrazole-4-carboxamide
N-(thiophen-2-ylmethyl)-1-(2-{[2-(trifluoromethyl)phenyl]formamido}ethyl)-1H-1,2,3-triazole-4-carboxamide
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-(3-chloro-2-fluorophenyl)-3-cyanopiperidine-1-carboxamide
N-[(2-methoxynaphthalen-1-yl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopropyl-3-{5-[(2,3-difluoro-6-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
ethyl 4-{[2-(dimethylsulfamoyl)ethyl]amino}piperidine-1-carboxylate
(3aS,6aR)-5-(5-hydroxypyrazine-2-carbonyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-(3-benzyl-1H-pyrazol-5-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine