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2-(cyclopropylmethyl)-8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(2-methoxyethyl)-2-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(methyl)amino)-1-phenylpropan-1-ol
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pent-4-enamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
ethyl 4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)benzoate
4-chloro-1,5-dimethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-3-carboxamide
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
(3S,4R)-1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[4-(4-{[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
2,7,8-trimethyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}quinoline-4-carboxamide
(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methanamine
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine
1-{4-[3-(2-methoxyphenoxy)azetidin-1-yl]piperidin-1-yl}ethan-1-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-hydroxy-N-(pyridin-3-ylmethyl)propanamide
1-(5-{[(3-fluorophenyl)methyl]amino}-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
5-[3-(2-methylphenyl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
1-[6-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-2-yl]ethan-1-ol
(1R,7S)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[(2-{5-[(4-methylphenyl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)methyl]-1λ6-thiolane-1,1-dione
N-cyclopentyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
7-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
3-[(3R,4S)-4-(dimethylamino)-1-[4-(hydroxymethyl)benzoyl]piperidin-3-yl]propan-1-ol
(3S,4R)-4-methyl-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-3-(2-methylpropyl)piperidin-4-ol
4-{1-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]piperidin-3-yl}benzoic acid
1-ethyl-N-{[3-(2-methoxyethoxy)phenyl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
(2S)-2-amino-N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-4-methylpentanamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
(1S,4S)-2-(4-chloro-2-methoxy-5-methylphenyl)-5-[2-(2,5-dimethoxyphenyl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
(2R)-N-(2,2-diphenylethyl)pyrrolidine-2-carboxamide
1-{[2-(2-chlorophenyl)phenyl]methyl}piperazine
4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl](pyridin-3-yl)methyl}morpholine
1-(1-{6-[4-(hydroxymethyl)-4-methylpiperidin-1-yl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
2-{methyl[2-(2-methylpiperidin-1-yl)ethyl]amino}propane-1,3-diol
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-4-yl)pyridine
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(hydroxymethyl)piperidin-4-ol
2-(dimethylamino)-N,4-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyrimidine-5-carboxamide
1-({1-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
(1S,5R)-3-[(2-chloro-5-fluorophenyl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)imidazolidin-2-one
N-(2-methylquinolin-4-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
5-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-(1H-imidazol-1-ylmethyl)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
N-(isoquinolin-5-ylmethyl)-N-methyl-3-(propan-2-yl)-1,2-oxazole-5-carboxamide