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2-(pyridin-4-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-amino-N,3-diethyl-N-(pyridin-4-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-[(3R,4S)-1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
7-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(1R,5R)-3-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
{1-[2-({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-2-yl}methanol
2-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-methyl-3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
4-(1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-3-yl)benzoic acid
2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]thiophene-3-sulfonamide
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
N1,N1-dimethyl-N3-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1,3-dicarboxamide
N-(pyridin-2-ylmethyl)-4-{[1-(pyridin-4-yl)piperidin-4-yl]oxy}benzamide
3,3,3-trifluoro-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
3-(pyridin-3-yl)-N-{[7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}propanamide
[(2,4-dimethoxyphenyl)methyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N,N-dimethyl-3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
2-(1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
9-[2-(3,4-difluorophenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-(4-{[(4-fluoro-3-methylphenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-methyl-5-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}pyrazine
1-{imidazo[1,2-b]pyridazine-3-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
methyl[3-(oxolan-2-yl)propyl](2-phenylethyl)amine
N-[2-(1H-indol-3-yl)ethyl]-2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(2-methoxyethyl)piperidine
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[2-(dimethylamino)ethyl]-N-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
1-{6-[4-(5-chloropyridin-2-yl)piperazin-1-yl]pyridin-2-yl}ethan-1-ol
4-[4-(1-benzyl-3-ethyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]pyridine
2-{[(5-butylthiophen-2-yl)methyl](methyl)amino}propanamide
3-(3-chloro-1,2-oxazol-5-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N,3,5-trimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzofuran-2-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
(2S)-4-(methylsulfanyl)-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}butanoic acid
1-benzyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
3-[3-(2-methylphenyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-1,4-diazepane
N-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-1-(furan-2-carbonyl)piperidin-3-amine
4-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-methyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
ethyl 3-({4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]phenyl}formamido)propanoate
1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]propan-1-one
(3aR,5S,6S,7aS)-2-({4-[methyl(phenyl)amino]phenyl}methyl)-octahydro-1H-isoindole-5,6-diol
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
1-{4-[2-(2,5-dihydro-1H-pyrrol-1-ylmethyl)phenoxy]butyl}-1H-imidazole
(2R,6R)-4-[4-(1H-pyrazol-4-yl)butanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid