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1-(1-methyl-5-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
3-({4-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)benzonitrile
6-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}-1,4-oxazepan-6-ol
1-ethyl-8-[3-(5-methylfuran-2-yl)butyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-4-methyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine-3,4-diol
3-methyl-3-[3-(oxolan-2-yl)propyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
methyl 7-oxo-9-[3-(pyridin-4-yl)propoxy]-3-(thiophene-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[2-(propylsulfanyl)phenyl]urea
4-[1-(3-methylbutyl)-5-(5-phenyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
(2R,6S)-2,6-dimethyl-4-{1-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}morpholine
1-(2-methanesulfonylethyl)-5-[4-(methylsulfanyl)phenyl]-4-phenyl-1H-imidazole
ethyl 4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]piperazine-1-carboxylate
1-benzyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}piperidin-4-amine
1-[(6-chloropyridin-3-yl)methyl]-4-(5-methyl-1-benzofuran-2-carbonyl)piperazine
N-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(pyridine-4-carbonyl)piperidin-4-amine
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-methylfuran-3-carboxamide
1-ethyl-4-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-1H-indole
(3-{2-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-(2-ethoxyethyl)-1-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N,N-diethyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1,8-dibenzyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]cyclopropane-1-carboxamide
2-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-3-[4-(2-methylpropyl)phenyl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[3-(4-fluorophenyl)phenyl]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(dimethylamino)propanamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl]propanoic acid
2-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]benzamide
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,2,3,6-tetrahydropyridine
6-(3-chlorophenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(3-methylbut-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(3S,4R)-3-acetamido-N-[(2-fluorophenyl)methyl]-4-(4-methylphenyl)pyrrolidine-1-carboxamide
N-{1-oxaspiro[4.5]decan-3-yl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
2-(1-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}piperidin-2-yl)acetic acid
3-methyl-4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)(pyridin-4-ylmethyl)amine
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
[(4S)-5-(4-acetyl-4-phenylpiperidin-1-yl)-4-amino-5-oxopentyl]urea
1,4-dimethyl-9-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4,9-triazaspiro[5.5]undecane
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(3-methylpyridin-4-yl)piperazine
1-(pyridin-3-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
N-cyclopropyl-1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-[(4aR,7aS)-6,6-dioxo-4-(pent-2-yn-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-(2-methoxyethyl)-1-methyl-N-(thiophen-2-ylmethyl)-1H-indazole-3-carboxamide
(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylpiperidin-4-yl)methanol
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1,2-oxazol-5-ylmethyl)acetamide
N5-cyclopropyl-N6-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine