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1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
1-[(2-methoxy-3,5-dimethylphenyl)methyl]-4-[2-(methylsulfanyl)ethyl]piperazine
4-[(4-fluorophenyl)methyl]-1-(1-methyl-1H-imidazole-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
9-(1-methyl-1H-pyrrole-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-(3-hydroxypyridine-2-carbonyl)-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
{4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-1-methylpiperazin-2-yl}methanol
4-{1-cyclohexyl-5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-1H-1,2,4-triazol-3-yl}pyridine
6-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5R)-6-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-butyl-4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
4-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
N-methyl-3-(N-methyl-1-{2-methylimidazo[1,2-a]pyridin-6-yl}formamido)butanamide
N-cycloheptyl-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carboxamide
6-(1-methyl-1H-pyrazol-4-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
4-(1H-imidazol-2-yl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
2-(dimethylamino)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(4-methylphenyl)acetamide
N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(5-phenyl-1,2-oxazole-4-carbonyl)piperazine
2-(2H-indazol-2-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)[(2E)-2-methylpent-2-en-1-yl]amine
4-{4-[(adamantan-2-yl)amino]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
ethyl 2-[4-(pyrimidin-5-ylmethyl)piperazin-1-yl]pyridine-3-carboxylate
2-{[(2-ethoxypyridin-3-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
3-[2-(4-phenyl-1H-imidazol-5-yl)-1H-pyrrol-1-yl]pyridine
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-6-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-acetyl-3-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
3-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
3-methyl-5-{4-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}-4H-1,2,4-triazole
1-{2-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
1-benzyl-N,2-dimethyl-5-(2-methylpropanamido)-N-[2-(oxan-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
8-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-ethylpiperidin-4-yl)-1-methyl-6-oxo-N-[2-(pyridin-2-yl)ethyl]-1,6-dihydropyridine-3-carboxamide
5,6-dimethyl-2-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
1-(furan-2-carbonyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
3,5-dimethyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1,2-oxazole-4-carboxamide
1-[4-(3,3-diphenylpiperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
4-ethyl-3-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-2H-1,2,3,4-tetrazole
3-(dimethylsulfamoyl)-N-methyl-5-[(2-methylpropyl)amino]-N-[1-(pyridin-2-yl)ethyl]benzamide
2-methyl-4-[4-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenyl]butan-2-ol
ethyl 4-(3-{[3-(1H-pyrazol-1-yl)phenyl]carbamoyl}piperidin-1-yl)piperidine-1-carboxylate
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
5-[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1,2,3-thiadiazole
9-methoxy-4-(3-methoxybenzoyl)-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine-1-carboxylate
1-(2-methoxyphenyl)-4-({2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
1-{4-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]-1,4-diazepan-1-yl}ethan-1-one