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1-(5-methyl-1H-pyrazole-3-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
4-[(5-chlorothiophen-2-yl)methyl]-1-(1H-indazol-6-yl)-5-methylpiperazin-2-one
1-{1-[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-methylpropan-2-yl}piperidine
3-[(3R,4S)-4-(dimethylamino)-1-[4-(methylsulfanyl)benzenesulfonyl]piperidin-3-yl]propanoic acid
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-methyl-3-[3-(1H-pyrazol-5-yl)phenyl]pyrazin-2-amine
5-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-2-methylpyrimidine
1-[(3,5-dimethylphenyl)methyl]-4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-2-one
1-[cyclohexyl(methyl)amino]-3-(2-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
7-chloro-4-[3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-[(2-butyl-1H-imidazol-4-yl)methyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
3-methyl-3-(1-methylpiperidin-4-yl)-1-[4-(pyridin-3-yloxy)phenyl]urea
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-amine
(1r,4r)-4-[({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]cyclohexan-1-ol
4-[2-(2-methyl-5-oxo-4-phenylpiperazin-1-yl)-2-oxoethyl]-1,2,3,6-tetrahydropyridazine-3,6-dione
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[2-(methylsulfanyl)ethyl]benzamide
N-cyclopentyl-1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine-4-carboxamide
2-methyl-N-[(1-propylpiperidin-3-yl)methyl]-3-[(pyridin-3-ylmethyl)amino]benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
3,5-dimethyl-4-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-2-yl)-1,2-oxazole
4-({2-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-[4-(2H-1,3-benzodioxol-5-yl)phenyl]-2-methyl-3-(2H-1,2,3,4-tetrazol-5-yl)pyridine
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
3-{5-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
(1S,5R)-3-(oxan-4-yl)-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1H-1,2,3-benzotriazole-5-carboxamide
3-[3-(4-methanesulfonylphenyl)phenyl]-1-(pyrrolidin-3-ylmethyl)-1H-pyrazole
3-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}benzonitrile
2-(4-hydroxyphenyl)-N-({1-[(3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
(1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}pyrrolidin-3-yl)methanamine
2-{[4-(2-phenylphenyl)piperazin-1-yl]methyl}pyridine-3-carboxylic acid
5-methyl-3-{3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}-1,2,4-oxadiazole
N-(5-cyanopyridin-2-yl)-4-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)benzamide
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azonane
N-methyl-N-(2-phenyl-1-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}ethyl)thiophene-3-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-(ethylsulfanyl)-5-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]pyrimidine
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-ol
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methylquinolin-6-yl)acetamide
(3aS,6aS)-2-[(1-benzyl-1H-indol-6-yl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide