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4-(2-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}ethyl)benzene-1-sulfonamide
N-{2-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethyl}acetamide
N,N-diethyl-5-[1-(5-methoxyfuran-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-[(3-methylphenyl)sulfanyl]piperidine
methyl 5-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
11-{[(2-chlorophenyl)methyl]amino}-4-[(2-fluorophenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}piperidin-4-yl)piperidin-4-ol
1-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
N-{2-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]ethyl}-N-methylmethanesulfonamide
6-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2,4-dimethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
(4aS,8aR)-6-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
5-ethyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1,2-oxazole-4-carboxamide
[(2,6-difluorophenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
(1R,5S,8S)-N-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
N2,N2,5,6-tetramethyl-N4-[(3-methylpyridin-2-yl)methyl]pyrimidine-2,4-diamine
(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-(1-{1-[(3-chloro-2,6-difluorophenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
9-(6-oxo-1-propylpiperidine-3-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
1-ethyl-3-(pyrrolidine-1-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-[(2-fluorophenyl)methyl]-2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
2-(3,3-diethylpyrrolidin-1-yl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
1'-(2-fluoro-4-methylbenzoyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{imidazo[1,2-a]pyridin-2-ylmethyl}acetamide
methyl 2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-6-(pyridin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(3-methyloxetane-3-carbonyl)pyrrolidine-3-carboxylic acid
methyl 5-[(4-hydroxybutan-2-yl)amino]-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(butan-2-yl)({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(thiophen-3-ylmethyl)amine
1-[(4-fluorophenyl)methyl]-4-(3-methyl-1,2-oxazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
methyl 3-[2-(4-fluorophenyl)acetyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(3-methylphenyl)methyl]-4-(pyrrolidin-3-ylmethyl)piperazine
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
methyl (2S,4R)-4-(dimethylamino)-1-[(2,4-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
4-(2-methoxy-4-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
3-[1-(5-cyanopyridin-2-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-(3-hydroxyphenyl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
N-methyl-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
N-(5-propyl-1,3,4-thiadiazol-2-yl)-2-[4-(pyrimidin-2-yloxy)piperidin-1-yl]acetamide
1-(2,2-difluoroethyl)-3-(2-methylphenyl)pyrrolidin-3-ol
(3S,4S)-1-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4-(dimethylamino)pyrrolidin-3-ol
5-benzyl-1-(3-methoxyphenyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-one
2-(dimethylamino)-7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(1-benzofuran-2-yl)-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
N-(1,4-dioxan-2-ylmethyl)-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
{1-[3-(hydroxymethyl)-4-methoxyphenyl]-1H-1,3-benzodiazol-2-yl}methanol
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(3-phenylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
dimethyl({5-[4-(4-methylbenzenesulfonyl)piperazine-1-carbonyl]-1,3,4-oxadiazol-2-yl}methyl)amine
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide