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N-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-chloro-5-(piperidine-1-carbonyl)phenyl]-3-(thiophen-3-ylmethyl)urea
2-cyclopropyl-8-[(1-ethyl-1H-indol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(pyridin-3-yl)-N-[(1r,4r)-4-methoxycyclohexyl]propanamide
5-cyclobutyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
4-(4-methylphenoxy)-1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidine
2-(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-2-yl)pyridine
methyl 3-({2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)propanoate
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrrolidin-2-one
5-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-2-(2-methoxyphenyl)pyrimidine
ethyl 4-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]piperidine-1-carboxylate
1-[4-({methyl[1-(2-phenylethyl)piperidin-3-yl]amino}methyl)thiophen-2-yl]ethan-1-one
5-chloro-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2,3-dihydro-1H-indole-2-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(quinoline-8-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(adamantan-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
2-methoxy-6-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-[(5-methylpyrazin-2-yl)methyl]-8-(1,2-oxazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(4-chlorophenyl)methyl]-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
1-{3-[3-(6-phenylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
1-[(2-chlorophenyl)methyl]-6-methyl-3-{[(thiophen-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-(3-methylpentan-3-yl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
(3S,4R)-1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
4-(hydroxymethyl)-1-[(2-phenylphenyl)methyl]azepan-4-ol
3-(1H-indol-3-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
8-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
(1R,3S)-N1-(2H-1,3-benzodioxol-5-ylmethyl)-N3-ethyl-1,2,2-trimethylcyclopentane-1,3-dicarboxamide
N-(2,3-dihydro-1H-inden-1-yl)-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{4-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]piperidin-1-yl}ethan-1-one
1-benzyl-N-ethyl-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
(2H-1,3-benzodioxol-4-ylmethyl)(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
N-[(2-chlorophenyl)methyl]-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
2-{4-benzyl-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{2-[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-(morpholin-4-yl)-2-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethan-1-one
2-(dimethylamino)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)acetamide
N-cyclohexyl-4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
(1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-(dimethyl-1,3-thiazol-5-yl)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]ethan-1-one
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-methoxy-5-(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyrimidine
8-[1-(2-chlorophenyl)piperidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-(3-methylphenyl)urea
2-(1-ethylpiperidin-4-yl)-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)ethan-1-one
6-fluoro-4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one