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4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-5-one
3-{3-ethyl-1-methyl-7-oxo-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-6-yl}azepan-2-one
3,5-dimethyl-1-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}azetidin-3-yl)-1H-pyrazole
[4-(2-amino-5,6-dimethylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
1-(2,4-dimethylphenoxy)-3-[(3-methylbutan-2-yl)amino]propan-2-ol
N,N-dimethyl-2-{2-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-1H-imidazol-1-yl}ethane-1-sulfonamide
3-[1-(5-acetylthiophene-2-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
(1S,5R)-6-(3-methyl-1,2-oxazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-benzyl-8-(1H-indol-3-ylmethyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
N-(3,4-difluorophenyl)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-amine
N-(1,3-dihydroxypropan-2-yl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
ethyl 4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-(3-methoxyphenyl)-4-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
(2S)-2-amino-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-phenylethan-1-one
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(methylsulfanyl)propan-1-one
3-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)-4H-chromen-4-one
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
{9-[3-(methylsulfanyl)propyl]-3-(thiophen-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]acetamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-1,2-dihydroquinolin-2-one
(1S,5R)-3-(2,8-dimethylquinoline-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]propane-1,2-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methylacetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
5-(2,2-diethylcyclopropanecarbonyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(2S,4R)-4-amino-N-ethyl-1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
2-(9-{[(3-fluorophenyl)methyl]carbamoyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetic acid
3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-amine
8-(2-aminopyridine-4-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N3,N5-dimethyl-4-oxo-1,N3-bis(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-cyclopentyl-9-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2,2-dimethylpropyl 9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate
(4aS,8aR)-6-(1H-1,3-benzodiazol-2-ylmethyl)-1-butyl-decahydro-1,6-naphthyridin-2-one
5-(4-fluoropiperidin-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(5-chloropyridin-2-yl)-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
methyl 4-[(3-aminopyrrolidine-1-carbonyl)amino]-2-chlorobenzoate
N-benzyl-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
N-(2,5-dimethylphenyl)-3-[(1-methyl-3-phenyl-1H-pyrazol-5-yl)formamido]propanamide
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
N-[2-(dimethylamino)ethyl]-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3R,4R)-1-(cyclopentylmethyl)-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-ethyl-1,2-oxazole-5-carboxamide
2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-methoxyethyl)-N,1-dimethyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(4-chlorophenyl)-2-[2-(1-ethylpiperidin-4-yl)acetamido]acetic acid