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4-ethoxy-1-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine
5-[(2-ethylpyrimidin-5-yl)methyl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-benzyl-3-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
3-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)-2,2-dimethylpropan-1-ol
N-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]methanesulfonamide
(2S,4R)-4-amino-1-(cyclohex-1-ene-1-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[5-(2,3-dihydro-1H-inden-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4,4,4-trifluorobutanamide
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
(2S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pentanamide
3-[(3-methoxyphenyl)methyl]-N-(thiophen-2-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(2-methoxyethoxy)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
(2R,3R)-3-(dimethylamino)-1'-[(trimethylpyrazin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-methyl-4-(piperidin-1-ylmethyl)-N-[1-(1,3-thiazol-5-yl)ethyl]benzamide
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
4-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
8-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}piperidin-3-yl)methyl]-1H-indole-2-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N,N,4-trimethyl-3-{[methyl(prop-2-en-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]propane-1,2-diol
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-ethoxypropan-1-one
4-ethyl-1-methyl-3-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxy-4-methylpentan-1-one
(3S,4R)-1-{[1-(2-carboxyethyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-(2-hydroxyethyl)-8-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(2S)-2-acetamido-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
4-({2-[1-(2,5-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-ethyl-6-(2-fluoro-3-methoxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
3-ethyl-6-(4-hydroxycyclohexyl)-1-methyl-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]azetidin-3-yl}piperidine
5-{2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-1,2,3,4-tetrazole
N-[2-(2-oxopiperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
3-[2-(ethylsulfanyl)phenyl]-1-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}urea
ethyl 2-[4-(1H-1,3-benzodiazol-2-ylmethyl)piperazin-1-yl]pyridine-3-carboxylate
8-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-4-({5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl}methyl)piperidine
1-(2,2-dimethylpropyl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
N-cyclopropyl-1-[(1s,4s)-4-(3-chlorobenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-chloro-2-methoxy-4-({[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amino}methyl)phenol
2-(4-chlorophenyl)-5-[1-(pyrimidin-4-ylmethyl)-1H-imidazol-2-yl]pyrimidine
1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-phenylpiperazine