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1-{2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-yl}piperidin-4-ol
(3aS,6aS)-2-(ethanesulfonyl)-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[(cyclopropylcarbamoyl)methyl]sulfamoyl}-N-(2,2,2-trifluoroethyl)benzamide
N-{1-[4-(dimethylamino)phenyl]-3-hydroxypropan-2-yl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(furan-2-ylmethyl)-1-(3-phenylpropyl)piperidin-3-amine
N-methyl-2-[methyl({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amino]acetamide
4-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]morpholine-2-carboxamide
1-{5-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-(methoxymethyl)-5-(3-propyl-1H-pyrazol-5-yl)-1,2,4-oxadiazole
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-indole-6-carboxamide
[(3-{4-azaspiro[2.5]octane-4-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)methyl]diethylamine
(3aR,5R,6S,7aS)-2-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-octahydro-1H-isoindole-5,6-diol
N-benzyl-N-methyl-1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidine-4-carboxamide
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-propoxypiperidine
1-[1-(6-cyanopyridine-3-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
4-chloro-1-methyl-3-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1H-indazole
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(morpholin-2-yl)ethan-1-one
5-{[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
4-[4-(2-methylphenoxy)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
2-(propan-2-yl)-8-(quinolin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(2-methyl-6-propylpyrimidin-4-yl)phenyl]ethan-1-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]-decahydro-1,6-naphthyridin-2-one
3-(propan-2-yl)-1-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}urea
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
N3-cyclooctyl-N5-ethyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-(thiophen-2-yl)urea
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N-ethyl-4-(4-methylpiperazin-1-yl)-N-(oxolan-2-ylmethyl)benzamide
3-{2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-oxoethyl}-4-[(4-phenylphenyl)methyl]piperazin-2-one
N-(2-fluorophenyl)-3-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)propanamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[2-(2-hydroxyethyl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
(3aR,6aR)-2-acetyl-5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[(3-hydroxyphenyl)methyl]piperazin-1-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
2-(1-ethylpiperidin-4-yl)-N-[furan-2-yl(phenyl)methyl]acetamide
2-[(furan-3-ylmethyl)(methyl)amino]-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
2-(2-hydroxyethyl)-8-[2-(phenylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
5-ethyl-4-({3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)furan-2-carboxamide
3-[2-(morpholin-4-ylmethyl)phenyl]benzonitrile
N-(6-cyanopyridin-3-yl)-4-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)benzamide
3-(5-methylthiophen-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
N-[(3R,4S)-1-[3-(dimethylamino)pyrazin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
1-(4-fluorophenyl)-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
N,N-diethyl-1-[(1s,4s)-4-(dimethyl-1,2-oxazole-4-sulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
N-benzyl{[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]amino}sulfonamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide