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4-methyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
2-oxo-N-[(1-phenylpiperidin-4-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
2-methyl-4-(2,3,4-trimethoxyphenyl)-1H-imidazole
1-methyl-4-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(propan-2-yl)piperazin-2-one
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2,6-dimethylquinoline-3-carboxamide
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-fluorophenyl)-N-(2-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
1-[3-(3-methoxyphenyl)phenyl]-3-methyl-3-(1-methylpyrrolidin-3-yl)urea
6-chloro-2-({4-[2-(furan-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}methyl)-1H-1,3-benzodiazole
4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}morpholine
N-(4-{[(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)carbamoyl]methoxy}phenyl)propanamide
2-hydroxy-5-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]benzamide
6-(3-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-N,N-dimethylpyridazin-3-amine
3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-(quinolin-6-yl)benzamide
N-(2,2-dimethyloxan-4-yl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
7-(2-hydroxyethyl)-6-oxo-N-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(3-methylpyridin-2-yl)-4-{[1-(trifluoromethyl)cyclopropyl]methyl}piperazine
2-[2-(1H-indol-3-yl)pyrimidin-5-yl]-N,N-dimethylquinoline-4-carboxamide
N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(1-methylpyrrolidin-2-yl)methyl]butanamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[2-(piperidin-1-ylmethyl)phenyl]urea
4-({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperazin-2-one
5-ethyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
4-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethylphenol
(4aR,7aS)-1-propyl-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-2-amino-N-butyl-N-(furan-2-ylmethyl)-3-(1H-imidazol-4-yl)propanamide
N-{1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-oxopropan-2-yl}methanesulfonamide
2-hydroxy-N-(1-methyl-1H-indazol-5-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
8-fluoro-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]quinoline-2-carboxamide
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[(4-fluorophenyl)methyl]-4-(3-methyl-1H-pyrazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
5-fluoro-2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
2-methyl-4-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)-6-(pyrrolidin-1-yl)pyrimidine
2-{5-[(2S)-2-amino-1-phenylpropan-2-yl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
8-[3-(3-methoxyphenyl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(2,6-difluoro-3-methylphenyl)methyl]-2-(4-methanesulfonylphenyl)-1H-imidazole
(2S,4R)-N-ethyl-4-{[(4-phenylphenyl)methyl]amino}-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
1-[3-(1H-indol-4-yl)phenyl]ethan-1-one
8-(5-methyl-1,2-oxazole-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,N-diethyl-1-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
5-[2-(3-fluorophenyl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
4-{2-oxo-2-[3-(1H-pyrazol-3-yl)piperidin-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
ethyl 1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
3-[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
N-(isoquinolin-5-ylmethyl)-N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-[(3R,4S)-4-cyclopropyl-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-3-yl]propanamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(3-hydroxy-3-methylbutyl)-N-methyl-1H-pyrazole-3-carboxamide
1-(furan-3-carbonyl)-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepane-6-carboxylic acid