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(4-{[methyl({5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl})amino]methyl}oxan-4-yl)methanol
1-(1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-2-phenylethan-1-one
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-[1-(4-fluorophenyl)propyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-(2,3-difluorophenoxymethyl)-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1,3-oxazole-4-carboxamide
4-chloro-N-methyl-N-(pyrazin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{9-[2-(2,3-dimethylphenoxy)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-N'-(2-fluoro-5-methylphenyl)butanediamide
3-(4-methoxyphenyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
5-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-2-(2-phenylethyl)-1,3-benzoxazole
2-(methylsulfanyl)-5-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)pyrimidine
N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-cyclobutanecarbonyl-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
6-(2-ethylmorpholin-4-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
4-benzyl-2-{2-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-methoxy-N-{[1-(quinolin-2-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
[(2-chloro-3,4-dimethoxyphenyl)methyl]({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
5-chloro-6-{2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxylic acid
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
2-(3-hydroxypropyl)-9-(3-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({5-[(4-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-3-carboxamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2,6-dimethoxybenzamide
2-{5-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-3-methylpyridine
dimethyl(3-{2-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-[9-(2,6-dimethylpyridin-4-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-[2-(benzyloxy)ethyl]-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-1-benzothiophene-5-carboxamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]quinoxaline-6-carboxamide
3-methyl-7-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(3-hydroxyquinoxalin-2-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)propanamide
2-{1-[(4-fluorophenyl)methyl]-4-(1H-indol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-[2-(2-methylphenyl)pyrrolidin-1-yl]acetamide
2-acetyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
3-{[1-(2-methoxyethyl)-3-(4-methyl-1,4-diazepane-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-indole
N-(2-hydroxyethyl)-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(propan-2-yl)propanamide
5-methyl-3-[3-(1H-pyrazol-3-yl)phenyl]-1,2,4-oxadiazole
6-methoxy-1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-indole-2-carboxamide
1-(1-benzofuran-3-carbonyl)-4-[(3-chlorophenyl)methyl]piperazine
5,6-dimethyl-N-[1-(thian-4-yl)piperidin-4-yl]pyridine-3-carboxamide
(1S,5R)-6-(3-fluoropyridine-4-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-[(2S)-1-benzylpyrrolidin-2-yl]-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazole
2-(9-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
[(5-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-chloro-4-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)phenol
N-(2-{1-[(2-phenylphenyl)methyl]piperidin-2-yl}ethyl)acetamide
2-(2-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one