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1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1'-[3-(piperidin-3-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
3-methyl-6-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyridazine
2-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
1-(1,2-oxazole-3-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-{[3-(methylsulfanyl)phenyl]methyl}-3-phenylpyrrolidin-3-ol
5-(azepane-1-carbonyl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(3,4-dichlorophenyl)-N,N-dimethylmorpholine-4-sulfonamide
(3R)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
methyl(4-{5-[(2E)-pent-2-en-3-yl]-4-phenyl-1H-imidazol-1-yl}butyl)amine
(1R,5R)-N,N-dimethyl-6-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[4-(3-ethenylphenyl)-1H-1,2,3-triazol-1-yl]methyl}cyclohexan-1-ol
8-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-N-(propan-2-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1R,9aR)-1-{[2-(methoxymethyl)-5-methyl-1H-1,3-benzodiazol-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-[(1-methylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(2-methylnaphthalen-1-yl)-1-[3-(methylsulfanyl)propyl]-1H-1,2,3-triazole
7-(2-methylphenyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-chloro-N,6-dimethyl-N-[1-(pyridin-3-yl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
(1S,5R)-6-(4-chlorobenzoyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}isoquinoline
4-methyl-2-{[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]methyl}-6-(trifluoromethyl)pyrimidine
(1-{2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
(1S,5R)-6-(cyclobutylmethyl)-3-{2-[4-(hydroxymethyl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
{2-fluoro-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]phenyl}methanol
2-{[(3,4-dichlorophenyl)methyl]amino}-N-(pyrazin-2-yl)acetamide
1-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-1,2-dihydroquinolin-2-one
7-[3-(piperidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
8-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[7-(cyclohex-3-en-1-ylmethyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenoxypropanamide
1-[(4-fluorophenyl)methyl]-4-(5-fluoropyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
methyl 6-(pyridin-3-ylmethyl)-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-benzyl-3-methyl-4-(pyridin-4-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
diethyl({2-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl})amine
(4aR,7aS)-1-{2-[methyl(pyridin-3-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-(oxan-4-yl)piperidine-4-carboxamide
3-{[bis(2-hydroxyethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
N-[4-(1H-pyrazol-1-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidine-2-carboxamide
ethyl 1-(cyclopentylmethyl)-3-(2-methoxyethyl)piperidine-3-carboxylate
1-(2-chloropyridin-3-yl)-3-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
2-cyclopentyl-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-ethyl-N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)pyrimidine-5-carboxamide
{[2-methoxy-5-(pyrimidin-5-yl)phenyl]methyl}(methyl)amine
dimethyl(2-{2-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
4-(4-fluorophenyl)-1-(pyrimidin-4-yl)piperidin-4-ol
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N6-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-N4,N4-dimethylpyrimidine-4,6-diamine