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1-(2-phenoxyethyl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazine
2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]-2-(thiophen-3-yl)acetic acid
N-[2-(azepan-1-yl)-2-phenylethyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-(2-methoxybutyl)benzamide
3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-N-(5-methyl-1,3-thiazol-2-yl)benzamide
6-[(diethylamino)methyl]-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(1-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(1-methyl-1H-imidazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-[(4aR,7aS)-4-[2-(2-methoxyethoxy)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(3aR,5S,6S,7aS)-2-{[2-(propylamino)pyrimidin-5-yl]methyl}-octahydro-1H-isoindole-5,6-diol
[(8-methoxyquinolin-2-yl)methyl](methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
1-(5-ethyl-1,2-oxazole-3-carbonyl)-2-(furan-2-yl)azepane
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
4-(4-acetyl-6-hydroxy-1,4-diazepane-1-carbonyl)-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
1-(3-methylbut-2-en-1-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)pyrrolidin-3-yl]acetamide
(3R,4R)-3-hydroxy-N-(2-methylphenyl)-4-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrrolidine-1-carboxamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,N,6-trimethylpyrimidin-2-amine
2-amino-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4-phenylpyrimidine-5-carboxamide
2-(azepan-1-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
3-[5-(1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[(2-methoxyphenyl)methyl]-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
2-(2-fluorophenyl)-5-(1H-imidazol-2-ylmethyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-methoxy-2-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
2-acetamido-N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)acetamide
(3S,4R)-N,N-dimethyl-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4-methylphenyl)pyrrolidin-3-amine
N-(2-methoxyethyl)-4-[6-(pyrrolidin-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[2-(ethylamino)ethyl]-1-[(3-methylphenyl)methyl]pyrrolidin-2-one
2-(4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)-N-(1-methyl-1H-pyrazol-5-yl)acetamide
4-(3-fluorophenoxy)-1-[2-(methylsulfanyl)benzoyl]piperidine
1-(3-methoxybenzoyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
1-[(3S,4R)-1-[2-(2H-indazol-2-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-2-(methoxymethyl)-6-methyl-1-(naphthalen-1-ylmethyl)-1,4-dihydropyridin-4-one
3-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(3-phenylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-amino-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-6-(2-methylpropyl)pyrimidine-4-carboxamide
5-(2-oxo-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)imidazolidine-2,4-dione
(1R,5S,8R)-3-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
2-(2-fluoro-3-methylphenyl)-2-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}acetic acid
9-[(1R,3S)-3-aminocyclohexanecarbonyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[1-(4-{7-methylthieno[3,2-d]pyrimidin-4-yl}phenyl)ethyl]morpholine
(1S,5R)-3-(2,6-dimethylpyrimidine-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(morpholin-4-yl)ethane-1,2-dione
2-chloro-N-({1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)pyridine-4-carboxamide
2-(2-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)pyridine
2-(phenoxymethyl)-N-[1-(pyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide