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N-[(5-chlorothiophen-2-yl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-ethyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-fluoro-N-(2-{[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridin-3-yl]formamido}ethyl)benzamide
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-(4-methylpiperazine-1-carbonyl)pyrrolidine-2-carboxylic acid
2-{4-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]piperazin-1-yl}pyridine-3-carbonitrile
ethyl 5-(5-methylpyrazine-2-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]urea
4-{2-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
(1R,7S)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
7-(2-methylphenyl)-4-[(3-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
4-(4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
(2R,4S)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-hydroxypiperidine-2-carboxylic acid
7-(1-benzothiophen-3-yl)-9-methoxy-4-propyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[5-cyclopropyl-4-(4-ethylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-[2-(trifluoromethyl)phenyl]pyrimidine
5-(2-methylphenyl)-3-(morpholin-4-yl)-1,2,4-triazine
3-(2,1,3-benzothiadiazol-5-ylmethyl)-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
2-methyl-3-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]pyridine
1-[4-(5-methylfuran-2-yl)benzoyl]-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
N-(1-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-phenoxyacetamide
1-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4-(furan-2-carbonyl)piperazine
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-3-(pyridin-3-yl)propanamide
N2-[1-(cyclohexylmethyl)piperidin-3-yl]pyrimidine-2,4-diamine
2-methoxy-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3,3,3-trifluoro-2-hydroxy-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
N-[(5-chlorofuran-2-yl)methyl]-N-(pyridin-3-ylmethyl)cyclopropanamine
2-benzyl-9-[3-(ethylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(3-chlorophenoxy)propan-1-one
8-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-ethyl-N-(2-hydroxyethyl)-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-(butan-2-yl)-7-{[(5-methylfuran-2-yl)methyl]sulfamoyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
({4-cyclopropyl-5-[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-{2-methyl-4-[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(1,1-dioxo-1λ6-thiolan-3-yl)benzamide
1-[(2-methoxyphenyl)methyl]-4-[4-(3-methylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(furan-2-yl)ethyl]-5-methoxybenzamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-methylbut-2-en-1-one
1-{2-hydroxy-3-[4-methoxy-2-(1,4-oxazepan-4-ylmethyl)phenoxy]propyl}piperidin-4-ol
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(9H-fluoren-2-ylmethyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)pyridin-2-amine
1-cyclooctyl-4-methyl-1,4-diazepan-5-one
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-(4-cyano-2-ethylphenyl)-4,4-difluoropiperidine-1-carboxamide
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-{1-imidazo[2,1-b][1,3]thiazol-6-yl-N-methylformamido}-2-(pyridin-3-yl)acetic acid
N-[(3R,4S)-1-benzyl-4-propylpyrrolidin-3-yl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide