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(2S)-N,1-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-(1-methanesulfonylpiperidin-4-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N,N-dimethyl-5-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(4-chlorophenyl)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
3-[5-(2,5-dimethylfuran-3-yl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
6-methyl-2-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}quinolin-4-ol
N-(2-ethoxybutyl)-2,6-dihydroxybenzamide
2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
(3S,4R)-4-methyl-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidine-3,4-diol
4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
1-cyclopentyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
1-[(6-chloro-2H-chromen-3-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
3-(2-oxoazepan-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
N-ethyl-6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxamide
4-{3-[1-(cyclopropylmethyl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylbenzamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propylsulfanyl)ethan-1-one
5-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-2-ol
8-(4-methoxy-2-methylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]quinoline
methyl({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
(3S,4S)-1-{5-amino-[1,2,4]triazolo[4,3-c]pyrimidin-7-yl}-4-cyclopropylpyrrolidine-3-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-(furan-2-ylmethyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(1-hydroxy-4-methylpentan-2-yl)-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-2,2-dimethylcyclopropane-1-carboxamide
3-(2-fluorophenoxy)-N-[4-methyl-3-(2-methylpropanamido)phenyl]azetidine-1-carboxamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
1-benzyl-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-amine
methyl 2-{1-[6-(methoxymethyl)pyrimidin-4-yl]pyrrolidin-3-yl}acetate
6-{[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]amino}pyridine-3-carbonitrile
2-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}pyrrolidine-1-carboxamide
(2S)-1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-2-(propan-2-yl)piperazine
3-[(3R,4S)-1-[(2-chloro-4-fluorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-N-(3-chloro-4-fluorophenyl)propanamide
4-ethyl-1-methyl-3-{[1-(3-phenoxypropanoyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[5-(2-ethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
2-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-{2-[2-(2-aminopyridin-3-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-2-(2-oxopyrrolidin-1-yl)propanamide
1-[(5-methylthiophen-2-yl)methyl]-3-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1-(pyridin-4-ylmethyl)urea
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
diethyl({5-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)amine
10-methoxy-5-[(1-methyl-1H-imidazol-5-yl)methyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)thiophene-3-carboxamide
1-[1-methyl-5-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)-1H-pyrrol-3-yl]ethan-1-one
2-{4-[3-(benzylsulfanyl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
2-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(oxan-2-ylmethyl)-3,4-dihydroquinazolin-4-one