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(2S,4S,5R)-2-ethyl-4-[(furan-2-ylmethyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
(2-methoxyethyl)({[4-(5-methylfuran-2-yl)phenyl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-(5,6-dimethylpyrimidin-4-yl)-N-(1-methyl-1H-indazol-5-yl)piperazine-1-carboxamide
N-[(3-fluorophenyl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carboxamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(4-fluorophenoxymethyl)-N-methyl-N-(2-phenylethyl)-1,3-oxazole-4-carboxamide
4-(4-fluorophenoxy)-1-(4-methylpyrimidine-5-carbonyl)piperidine-4-carboxylic acid
3-(5-{2-[2-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
1-[2-(naphthalen-1-yl)acetyl]-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(2-phenoxyethyl)piperazine
N-[(2S)-1-[(2S,4S)-2-{[(dimethylcarbamoyl)amino]methyl}-4-fluoropyrrolidin-1-yl]-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl]acetamide
1-(cyclopropanesulfonyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-[5-(3-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]-N-methylethane-1-sulfonamide
2-{2-[(5-methoxy-1-methyl-1H-indol-2-yl)formamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
4-cyclobutyl-6-methyl-N-(1-propylpiperidin-4-yl)pyrimidin-2-amine
3-hexyl-8-[2-(3-oxopiperazin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-cyclohexyl-2-(4,6-dihydroxypyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
N-(furan-2-ylmethyl)-9-methoxy-3-{[3-(2-methylphenyl)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}quinoline
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
N,N-dimethyl-3-[({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amino)methyl]pyridin-2-amine
5-[4-(cyclopentylmethyl)piperazine-1-carbonyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
4-[5-methyl-4-(4-methylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
1-[2-(cyclobutylformamido)ethyl]-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(azepan-1-yl)ethyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3,5-dimethyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]adamantane-1-carboxamide
2-{3-[({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}carbamoyl)amino]phenyl}acetamide
N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclohexyl-3-[2-(dimethylamino)-2-(2-fluorophenyl)acetamido]propanamide
1-{2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-oxoethyl}pyrrolidin-2-one
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
4-(2-amino-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)-N-methylbenzene-1-sulfonamide
(1R,5S)-6-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
methyl 1-benzyl-3-(oxolane-2-amido)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}butanamide
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}cyclopropane-1-carboxamide
3-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-ethyl-5-oxopyrrolidine-3-carboxamide
3-[5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-2-methoxyquinoline
2-(4-fluorophenoxymethyl)-4-hydroxy-N-[1-(pyrimidin-4-yl)ethyl]pyrimidine-5-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-6-methoxy-1-methyl-N-(prop-2-en-1-yl)-1H-indole-2-carboxamide
3-ethyl-6-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(3-fluorophenyl)ethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]methanol
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-[5-(thiophen-2-yl)furan-2-yl]propanamide
(3R)-3,4,4-trimethyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-ol
(1R,5R)-6-(cyclobutylmethyl)-3-(4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
[5-(dimethoxy-1,3,5-triazin-2-yl)-2-fluorophenyl]methanol