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N,N-dimethyl-4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazine-1-carboxamide
1-[2-(1H-indol-5-yl)pyrimidin-4-yl]piperidin-4-ol
(2R,3S)-N2-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-N3-(prop-2-en-1-yl)bicyclo[2.2.1]heptane-2,3-dicarboxamide
N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)-1H-indole-6-carboxamide
N-(3-methoxypropyl)-N-[(8-methoxyquinolin-2-yl)methyl]-1-methylpiperidin-4-amine
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropanesulfonamide
4-hydroxy-N-{2-[methyl(phenyl)amino]propyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
5-methyl-3-(3-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-3-oxopropyl)-2,3-dihydro-1,3-benzoxazol-2-one
(4S,4aS,8aS)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-phenyl-decahydroquinolin-4-ol
2-[(4aR,7aS)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
N-cyclopropyl-2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]pyridine-4-carboxamide
2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidine-1-carbonyl}pyrazine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)propanamide
4-(5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(1S,5R)-3-[4-(1H-indol-3-yl)butanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-({2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}formamido)ethyl]pyridine-3-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[1-(2-methoxyethyl)-7-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
2,6-dimethyl-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,4-dihydropyridin-4-one
N-methyl-N-[2-(methylamino)ethyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[4-(3-methoxypropyl)piperazin-1-yl]ethan-1-one
5-(3-acetylphenoxymethyl)-N-[2-(diethylamino)ethyl]-N-ethyl-1,2-oxazole-3-carboxamide
1'-[3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
ethyl 4-{2,8-diazaspiro[4.5]decan-2-yl}piperidine-1-carboxylate
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
4-{[(3S,4S)-3-hydroxy-4-[methyl(propyl)amino]pyrrolidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-(propan-2-yl)pyridine-4-carboxamide
2-oxo-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1,2-dihydroquinoline-4-carboxamide
5-(hydroxymethyl)-2-methyl-4-{[3-(thiophene-2-carbonyl)piperidin-1-yl]methyl}pyridin-3-ol
1-(furan-3-ylmethyl)-3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-(3-methoxypropyl)-1-[3-(trifluoromethyl)benzoyl]piperidine
6-[(diethylamino)methyl]-N-(2,6-dimethoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(5-methoxyfuran-2-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
2-(dimethylamino)-2-(4-methylphenyl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
N-(2-fluoroethyl)-3-{[3-oxo-3-(pyrrolidin-1-yl)propyl]sulfamoyl}benzamide
3-(2H-1,3-benzodioxol-5-yl)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
1-[2-(3-chlorophenyl)ethyl]-N-[2-(diethylamino)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(3S,4R)-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2-methyl-1,4-diazepan-5-one
1-{4-[(2-propoxyethyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-(4-methoxyphenyl)-2,2-dimethyl-4-(5-propyl-1,2-oxazole-4-carbonyl)piperazine
(3aR,7aS)-2-{2-[(2-methylpyrimidin-4-yl)oxy]hex-5-en-1-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(2S)-2-{[1-(4-fluorophenyl)cyclopropyl]formamido}-3-(pyridin-4-yl)propanoic acid
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(1S,5R)-6-(cyclobutylmethyl)-3-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,7aR)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-ol
2-(2-methoxyethoxy)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
4-hydroxy-N,N-dimethyl-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide