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6-[1-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
3-(3-{[(2-methanesulfonylethyl)amino]methyl}-1H-indol-1-yl)propanamide
2-amino-N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3S,4R)-3-benzyl-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-methylpiperidin-4-ol
N-(2-hydroxyethyl)-3-methoxy-2,2-dimethyl-N-[(2-methylphenyl)methyl]propanamide
8-(2-benzyl-1,3-thiazole-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
6-(2,5-dimethylfuran-3-yl)-2-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
(1R,9aR)-1-{3-[2-(methylsulfanyl)ethyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl}-octahydro-1H-quinolizine
5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,3-benzothiazol-2-amine
2-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-4-(3,3,3-trifluoropropyl)pyrimidine
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(2-{[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)carbamoyl]amino}phenyl)-N,N-dimethylpropanamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]benzamide
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
3-{1-[2-(methylamino)pyridine-4-carbonyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(diphenylmethyl)-N-ethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-cyclohexyl-3-phenylpropanamide
N6-(2-methoxyethyl)-N5-methyl-N5-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-ethyl-9-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(cyclopropylmethyl)-4-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-yl]ethan-1-ol
N-[(2,3-difluorophenyl)methyl]-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(2-oxoazepan-1-yl)acetamide
(4aR,7aS)-1-ethyl-4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{4-chloro-2-[4-(2-hydroxyethyl)piperazine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
N-[2-(morpholin-4-yl)ethyl]-4-(piperidin-3-yl)benzamide
4-[2-(piperidine-1-carbonyl)phenoxy]-1-(4,4,4-trifluorobutyl)piperidine
2-{2-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2,2-dimethyl-3-[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]propan-1-ol
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-oxo-2-(pyrrolidin-1-yl)acetamide
3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-(4-chloro-3-fluorophenyl)-3-methyl-3-[2-(2-oxopiperidin-1-yl)ethyl]urea
3-(1H-1,2,3-benzotriazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
1-(3-cyano-4,6-dimethylpyridin-2-yl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}piperidin-3-ol
(2S,4S)-1-(2,2-diphenylethyl)-N-methyl-4-{[(3,4,5-trimethoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-(4-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-(3-methyl-4-{[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
N-[(3-fluorophenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
1-(furan-2-ylmethyl)-4-[2-(1,3-thiazol-4-yl)acetyl]-1,4-diazepane-6-carboxylic acid
(2S,4S)-4-(2,2-dimethylpropanamido)-1-methyl-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidine-2-carboxamide
4-ethenyl-N-[2-(1-methylpiperidin-3-yl)ethyl]benzamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-(5-methyl-1H-pyrazol-1-yl)propanamide
(3aS,7aR)-5-methyl-2-[4-(propan-2-yloxy)benzoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-(methoxymethyl)-N-[3-(methylsulfanyl)propyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-(1-cyclopentanecarbonylpiperidin-3-yl)-4-(2-fluorophenyl)piperazine
N-[(1S)-2-hydroxy-1-phenylethyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide