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4-(2,3-dihydro-1H-isoindol-2-yl)-N-[3-(1H-imidazol-1-yl)propyl]pyridine-2-carboxamide
1-(4-fluorophenyl)-6,6-dimethyl-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-{[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}propan-1-ol
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[1-(4-methoxyphenyl)propyl]-N-methylacetamide
(3aR,6aR)-2-[2-(3,4-dimethylphenoxy)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-oxoethyl}-2,3-dihydro-1H-indazol-3-one
1-{1-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-yl}piperidine
4-hydroxy-1-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperidine-4-carboxylic acid
N3-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-N3-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
N-[(1-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-methyl-1H-indole-2-carboxamide
1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
5-[butyl(methyl)amino]-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-ethyl-N-(1-{1-[(4-methylphenyl)amino]cyclopentanecarbonyl}pyrrolidin-3-yl)acetamide
2-ethyl-4-phenyl-9-(pyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecane
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{6-chloro-3-[(4-methylpiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-[4-(3-cyanophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
methyl 2-{4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
1-{[(2R,5S)-5-[(1-methyl-1H-indazol-5-yl)methyl]oxolan-2-yl]methyl}piperidine-4-carboxylic acid
3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
(2S,3R)-2-amino-3-hydroxy-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
1-[1-(3,5-difluorobenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylamino)pyridine-4-carboxamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-ethyl-N-(2-methoxyethyl)butanamide
2-(3-chloro-2,6-difluorophenyl)-1-(furan-3-ylmethyl)-1H-imidazole
2,4-dimethoxy-6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1,3,5-triazine
1-[(5-ethylpyridin-2-yl)methyl]-3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]urea
{4-benzyl-1-[3-(3-fluorophenyl)benzoyl]piperidin-4-yl}methanol
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-2-(4-ethylpiperazin-1-yl)acetamide
8-(2,2-dimethylpropyl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(5-methylpyrazine-2-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
N-[(4-methylphenyl)methyl]-1-{2-[3-(pyridin-3-yl)propanamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-[(3-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]carbamoyl}phenyl)amino]acetic acid
2-[4-(1-benzyl-1H-pyrazole-4-carbonyl)-1-methylpiperazin-2-yl]ethan-1-ol
9-[(2-aminopyridin-3-yl)methyl]-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-methylbutanamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
4,4,4-trifluoro-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}butanamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
2-(3,5-difluorophenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
5-{3-[1-(dimethylamino)ethyl]phenyl}-1H-indazol-3-amine
1-[(3-methylphenyl)methyl]-4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-2-one
3-(hydroxymethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
3-[(3R,4S)-1-(4-methylphthalazin-1-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-[2-(3-fluorophenyl)ethyl]-6-methylpyrimidin-2-amine