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4-cyclopentyl-2-[4-(1H-imidazol-2-yl)piperidin-1-yl]pyrimidine
6-(2-fluoro-4-methoxyphenyl)-7-methyl-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-(4-benzyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(furan-2-yl)ethyl]acetamide
3-[(4aR,7aS)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-3,5-dimethyl-1H-pyrazole
4-(hydroxymethyl)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidin-4-ol
N,6-dimethyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(1H-pyrazol-1-yl)benzamide
3-[(propan-2-yl)({[(1s,4s)-4-aminocyclohexyl]methyl})amino]propanamide
2-[4-(2,4-difluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-{[7-(4-cyclopropanecarbonylphenyl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-3-carboxamide
2-{[2-(1H-imidazol-1-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-2-(2-oxopyrrolidin-1-yl)propanamide
(3S,4R)-1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-(4-methoxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
4-[1-(pyridin-3-yl)pentyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-4-methoxy-N-(2-methoxyethyl)benzamide
3-ethyl-8-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)pyrrolidin-2-yl]-1,3-benzothiazole
(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
1-(4-methoxyphenyl)-6,6-dimethyl-4-(quinolin-6-ylmethyl)piperazin-2-one
(3S,4S)-1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4-propylpyrrolidine-3-carboxylic acid
3-{2-[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
methyl 3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6,7-dimethoxy-2-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-7-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
(1R,3S)-3-(2-hydroxyethoxy)-7-(oxan-4-yl)-7-azaspiro[3.5]nonan-1-ol
N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]thiophene-2-carboxamide
1-[4-(3-acetylphenyl)phenyl]-3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-methylurea
3-phenyl-1-[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]propan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
3-[3-(dimethylamino)propyl]-5-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
2-{1-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(furan-2-ylmethyl)-N-methylacetamide
1-(1,3-benzothiazol-6-yl)-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)urea
2-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-2,8-diazaspiro[4.5]decane
(1S,5R)-6-(5-propylthiophene-3-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-methoxyethyl)-8-[2-(phenylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
6-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyridazin-3-amine
ethyl 3-{[4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]amino}propanoate
1-[4-(4-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-2-ethylbutan-1-one
N-methyl-N-(quinoxalin-2-ylmethyl)-1,3-thiazole-4-carboxamide
N-[(2R)-1-hydroxy-3-phenylpropan-2-yl]-3-(2-methyl-1H-indol-1-yl)propanamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(6-methylpyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
4-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
2-(2,4-dichlorophenoxy)-1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethan-1-one