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4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(thian-4-yl)benzamide
3-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
N-(2-methoxyethyl)-1-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-1-[(6-ethoxypyridin-3-yl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
6-[2-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidin-4-amine
({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)[1-(pyridin-4-yl)propan-2-yl]amine
5-{[benzyl(methyl)amino]methyl}-N-[(2,3-difluorophenyl)methyl]-1,2-oxazole-3-carboxamide
N3-[2-(3-fluorophenyl)ethyl]-N5-[(2-fluorophenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-benzyl-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,2-oxazole-5-carboxamide
{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
1-[(2-fluorophenyl)methyl]-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidin-3-amine
3-[({1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
5-{5-[(2S)-butan-2-yl]-1,2,4-oxadiazol-3-yl}-2-methanesulfonyl-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
(2H-1,3-benzodioxol-4-ylmethyl)({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
1-[3-(5-methylfuran-2-yl)butyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
benzyl({[4-(pyrimidin-5-yl)phenyl]methyl})amine
3-(3-fluoro-4-phenylbenzoyl)-1-(1H-imidazol-2-ylmethyl)piperidine
1-methyl-8-{6-methylthieno[2,3-d]pyrimidin-4-yl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methoxypyrazine
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
8-(6-fluoro-4-methylquinolin-2-yl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)-1,3-benzothiazole
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1,2-oxazole-3-carboxamide
(5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-propoxyphenyl)methanol
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
3-{[6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
5-benzyl-5-[1-(furan-3-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
2,5-dimethyl-3-{4-[2-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl}pyrazine
N-{2-[ethyl(3-methylphenyl)amino]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
2-(4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
3-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(4H-1,2,4-triazol-4-yl)ethyl]amino}methyl)piperidin-2-one
3-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}phenol
4-[1-(3-chlorothiophene-2-carbonyl)piperidin-3-yl]-5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidine
2-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)quinolin-4-ol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazol-5-yl}benzoic acid
N-cyclopropyl-2-({1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
1-ethyl-N-methyl-5-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxamide
3-ethyl-4-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-methyl-4-{[4-(2-phenylethoxy)phenyl]methyl}piperazine-2-carboxylic acid
1-{3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}piperazine
3-methyl-7-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide
1-(4,6-dimethylpyrimidin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-amino-N-[1-(3-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
1,N3-dibenzyl-N5-ethyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-hydroxy-N-[(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)methyl]pyridine-3-carboxamide