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3-(2-butylpyrrolidine-1-carbonyl)-5-(phenoxymethyl)-1H-pyrazole
(1S,2S)-2-{5-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-4-phenyl-1H-imidazol-1-yl}cyclohexan-1-ol
3-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-[(3-hydroxy-4-methoxyphenyl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-{3-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methylphenyl)propan-1-one
2-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carbonitrile
2-[1-(5-phenyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-(but-3-enoyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
2-(5-acetylthiophen-3-yl)-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]acetamide
1-{1'-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-ethyl-5-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyrimidin-2-amine
3-({2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}sulfonyl)benzoic acid
2-methoxy-3-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
1-{1-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]-1,2,3,6-tetrahydropyridin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2-ethoxyethyl)-N,3-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
8-[(3-methoxyphenyl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-4,6-dimethylpyrimidine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-{4-[3-(propoxymethyl)pyrrolidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}pyridine
4-[6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine-3-carbonyl]morpholine
4-(1,3-benzothiazole-6-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-(4-methyl-2-oxo-2H-chromen-7-yl)-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
1-[(5-ethylfuran-2-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-(2-methyloxane-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(4-fluorophenyl)-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]morpholine
6-methyl-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}-2-(ethylsulfanyl)pyrimidine
N-[(2,3-difluoro-4-methylphenyl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(2-fluorophenyl)methyl]-2-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]acetamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
4-[5-(2-methylpropyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
2-(dimethylamino)-N-{2-[4-(dimethylamino)phenyl]ethyl}-2-(3-fluorophenyl)acetamide
N-{[1-(methoxymethyl)cyclopentyl]methyl}-4-(piperidin-1-ylmethyl)benzamide
2-phenyl-5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyrimidin-4-ol
2-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylpyridine-3-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(2-methylbutanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-[(4-methylpiperazin-1-yl)sulfonyl]-2-(1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
3-hydroxy-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
3-(3-fluorophenyl)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
methyl 3-(2-methoxyacetamido)-5-{[(9-methyl-9H-carbazol-3-yl)formamido]methyl}benzoate
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-N-[(3-methyloxetan-3-yl)methyl]benzene-1-sulfonamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]propan-1-one
3-(2-methylpropyl)-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1,2-oxazole-5-carboxamide
N-[2-(2,3-dichlorophenyl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
1-(4-aminopyrimidin-2-yl)-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylic acid
3-[(4aR,7aS)-6,6-dioxo-4-[3-oxo-3-(pyrrolidin-1-yl)propyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-2-{4-[4-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}acetamide