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methyl 5-[(1-ethylpiperidin-4-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3-chlorophenyl)methyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
6-methyl-3-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-(pyridin-3-yl)acetamide
4-cyclopropyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-methyl-N-(oxan-3-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(2-methoxyethyl)-3-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}propanamide
3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-phenylpyrrolidin-2-one
2-[3-(3-acetamidophenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-{[6-(cyclohex-1-en-1-yl)pyridin-3-yl]methyl}-4-methylpiperazine
N-({1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
(2S,4S)-4-amino-N-methyl-1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}pyrrolidine-2-carboxamide
5-[4-(azepane-1-carbonyl)-3,6-dimethylquinolin-2-yl]pyrimidin-2-amine
1-{[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
4-({1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}oxy)benzoic acid
8-(5-acetylpyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-2,1,3-benzoxadiazole
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]propanamide
8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-2,2-dimethyloxan-4-amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
N'-(2,4-dimethylphenyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]ethanediamide
2-{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}-1,3-benzoxazole
5-(2-chlorophenyl)-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]furan-2-carboxamide
{2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
2-(2,4-dichlorophenoxy)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
1-(cyclobutylmethyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(5-methyl-1,2-oxazol-3-yl)-N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]pyrrolidine-1-carboxamide
2,6-dimethyl-4-[({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]phenyl acetate
3-chloro-4-{[1-(2-hydroxyethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N,N-dimethyl-5-(1-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)-1,3-thiazol-2-amine
1-(4-chloro-3-fluorobenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
ethyl 2-(1-{2-[4-(pyridine-2-amido)-1H-pyrazol-1-yl]acetamido}cyclohexyl)acetate
2-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amino}methyl)-4-fluorophenol
2-(2-phenylethyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
6-methoxy-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carbonitrile
2-(2-ethoxyethyl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
3-ethoxy-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-methyl-N-[({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}carbamoyl)methyl]propanamide
6-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidin-4-amine
3-(2-methoxyphenyl)-N-[1-({[1-(naphthalen-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
N-methyl-N-[(3-methyloxetan-3-yl)methyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyrrolidin-1-yl)benzamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
8-[4-(2-methoxyphenyl)benzoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N,N,8-trimethyl-2-{2-[(pyridin-4-ylmethyl)amino]pyrimidin-5-yl}quinoline-4-carboxamide
N-[(1-methylpiperidin-3-yl)methyl]-2-(propylsulfanyl)acetamide