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5-fluoro-N,N-dimethyl-2-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyrimidin-4-amine
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-methylbutyl)propanamide
3-[2-(4-methoxyphenyl)ethyl]piperidine
2-[(3,4-difluorophenyl)methyl]-8-[2-(dimethylamino)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
N-[1-(4-hydroxyphenyl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-(2-{1-[(3-chlorophenyl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl}ethyl)acetamide
5-ethyl-N-methyl-N-[2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
4-benzyl-1-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]piperidin-4-ol
2-{1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-2-yl}-1-methyl-1H-1,3-benzodiazole
(2S,4R)-4-amino-1-[2-(phenylformamido)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4,4,4-trifluoro-1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
3-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)propan-1-ol
1-(2-{[(1,3-benzoxazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
N-(3-cyano-4-ethoxyphenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-(3-methylbutyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(2H-1,3-benzodioxol-4-ylmethyl)[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amine
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
7-[(4-benzoylpiperazin-1-yl)methyl]-4-methyl-2H-chromen-2-one
methyl 5-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-5-oxopentanoate
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[(6-hydroxypyrimidin-4-yl)methyl]butanamide
N,2-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[(3R,4S)-1-[(3-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
6-ethyl-2-(morpholin-4-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-4-amine
N-[2-(4-chlorophenyl)ethyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
1-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-imidazole-4-sulfonamide
3-{1-[(4-fluorophenyl)methanesulfonyl]piperidin-3-yl}benzoic acid
5-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
3-butyl-4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1-methylpiperazin-2-one
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
(1S,2R)-N2-tert-butyl-N1-(2-carbamoylethyl)-N1-(propan-2-yl)cyclohexane-1,2-dicarboxamide
6-(3-carbamoylpiperidin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
2-methyl-8-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)ethan-1-one
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
4-methyl-2-(3-phenyl-5-{[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazol-1-yl)pyridine
4-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
2,5,6-trimethyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrimidin-4-amine
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-phenyl-1,2-oxazole
2-[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]benzene-1,3-diol
3-{[1-(2-chlorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
2-[2-(1H-imidazol-1-yl)ethyl]-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
3-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)-6-methyl-4H-chromen-4-one
8-(2,3-dihydro-1H-inden-2-yl)-3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione