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3-(4-{imidazo[1,2-a]pyridine-3-carbonyl}piperazin-1-yl)-1-azabicyclo[2.2.2]octane
2-{2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]ethyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-methyl-2-(4-methyl-1,4-diazepan-1-yl)-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-(4-fluorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)propanamide
1-{3-oxo-3-[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
6-butyl-2-(2-{[3-(dimethylamino)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-ethyl-5-{[methyl(2-phenylethyl)amino]methyl}-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-(2-methoxy-4-methylbenzenesulfonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-[2-methoxy-4-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-[3-(3-methoxypyrrolidine-1-carbonyl)benzenesulfonyl]piperidine-4-carbonitrile
6-[(3,5-dimethoxyphenyl)methyl]-1-(4-methyl-1,4-diazepane-1-carbonyl)-6-azaspiro[2.5]octane
({4-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
2-amino-4-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
8-(4-aminocyclohexyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(4-chloro-2-fluorophenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
8-[(2,6-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-(2H-1,3-benzodioxol-5-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(2-ethoxyphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-2-(pyridin-3-yl)quinoline
8-{[4-(1-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinoline
3-[3-(3-hydroxypiperidin-1-yl)propyl]-1-[2-(pyridin-2-ylmethoxy)phenyl]urea
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
6-{[(1-ethyl-1H-imidazol-5-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1,9-dimethyl-4-[4-(1H-pyrazol-4-yl)butanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
6-[(oxolan-2-ylmethyl)sulfamoyl]-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-methyl-2-(methylsulfanyl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
3-(1H-indol-3-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2-methylphenyl)methyl]piperidin-4-yl}oxy)benzamide
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[3-(pyridin-4-yl)propyl]pyrrolidin-2-one
1-(4-chlorophenyl)-N-[(4-hydroxyazepan-4-yl)methyl]cyclohexane-1-carboxamide
4-ethyl-6-{4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}pyrimidine
3-(2-fluoro-5-methoxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
5-methyl-1-(2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(3,5-dimethylphenyl)methyl]-4-(4-methylpyrimidine-5-carbonyl)piperazin-2-one
N-(3-chloro-4-fluorophenyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
3-(1H-pyrazol-1-yl)-N-[3-(pyridin-3-yloxy)propyl]benzamide
N-[2-(1H-imidazol-4-yl)ethyl]-3,5,7-trimethyl-1H-indole-2-carboxamide
1-benzyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-4-(2,5-dimethylthiophen-3-yl)pyrimidine
(3R,5S)-N3-(4-fluorophenyl)-1-[(4-hydroxyphenyl)methyl]-N5-(naphthalen-1-ylmethyl)piperidine-3,5-dicarboxamide
3-benzyl-1-methyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(2-methoxy-5-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-5-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,4-triazole