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2-(5-chloro-2-methoxypyridin-4-yl)-5-fluoro-4-methoxypyrimidine
ethyl 4-[2-chloro-5-(1H-pyrazol-1-yl)benzamido]piperidine-1-carboxylate
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(2-phenylethyl)pyrrolidin-3-yl]methanol
1-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-3-yl)-4-(2-fluorophenyl)piperazine
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethoxyethan-1-one
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-indole
1-(cyclopent-1-ene-1-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
3-fluoro-N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-4-(1H-1,2,4-triazol-1-yl)butanamide
(5S,9aS,9bS)-5-(isoquinolin-5-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(2-fluorophenoxy)-1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)azetidine
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-[(2-methylpyridin-3-yl)oxy]-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-4-methylpyrimidine-5-carboxamide
6-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidine-1-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
1-[(5-acetylthiophen-3-yl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
4-(1H-indazol-5-yl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
N,N-dimethyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridine-3-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
7-(3-chlorophenyl)-4-(2-methylpyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclopropyl-2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[(3-methylthiophen-2-yl)methyl]acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(methylsulfanyl)benzoyl]pyrrolidine-3-carboxylic acid
N,2,7,8-tetramethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}quinoline-4-carboxamide
2-{2-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1-methyl-1H-1,3-benzodiazole
3-methyl-4-({[2-(5-methylfuran-2-yl)ethyl]carbamoyl}amino)-N-propylbenzamide
methyl 4-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}benzoate
1-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-2-phenylethan-1-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(hydroxymethyl)benzoyl]pyrrolidine-3-carboxylic acid
6-chloro-3-{[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4H-chromen-4-one
1-[(2,6-difluorophenyl)methyl]-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
2-(4-chloro-2-methylphenoxy)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
1-cyclopentanecarbonyl-N-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidine-4-carboxamide
N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
3-{[(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1'-(3-ethoxybenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(4-fluorophenyl)methyl]-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
ethyl 5-(3-methyl-4-oxo-3,4-dihydrophthalazine-1-carbonyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
7-(2,4-dimethylbenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-(1H-imidazole-5-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
N-ethyl-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
2-(2-aminoethyl)-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
(2S,4R)-4-amino-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})(pyridin-3-ylmethyl)amine
N-methyl-5-[(5-phenylthiophen-2-yl)methyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
(5S,9aS,9bS)-5-(3-fluorophenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(2,3-dimethoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one