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N-[2-oxo-4-(2-propylpyrimidin-5-yl)-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
7-(3-chlorophenyl)-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(cyclohexylmethyl)-6-oxo-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
5-{[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N,2-dimethyl-N-(2-phenylethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]quinoxaline
(3S,4S)-1-(butane-1-sulfonyl)piperidine-3,4-diol
4-{[2-(dimethylamino)-2-(2-fluorophenyl)acetamido]methyl}benzoic acid
1-[1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-4-yl]piperidin-3-ol
N-[2-(pyridin-3-yloxy)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylfuran-2-carboxamide
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
2-(methylamino)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1,3-thiazole-4-carboxamide
9-(3-hydroxy-4-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-aminoethyl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{1-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1H-imidazol-2-yl}benzoic acid
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperazine
2-{2-[2-(3-methoxyphenyl)piperidin-1-yl]ethoxy}ethan-1-ol
(1S,6R)-9-(2-methoxypyridine-4-carbonyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
{[3-(3-methoxyphenyl)oxolan-3-yl]methyl}(2-methylpropyl)(pyridin-2-ylmethyl)amine
3,5-dimethyl-4-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1,2-oxazole
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-propyl-1H-pyrazole-5-carboxamide
N-({7-[(2-hydroxy-3-methoxyphenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
2-[(3-carboxypropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(2S)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-3-carboxamide
2-methyl-5-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-{3-[(3,5-dimethoxyphenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperidine
(5S,9aS,9bS)-5-(6-chloro-2H-1,3-benzodioxol-5-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[(4-acetylpiperazin-1-yl)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
N-(2,4-dimethoxyphenyl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propanamide
2-phenoxy-N-{[7-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
3-chloro-N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
3-[(3-fluorophenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(5-propyl-1,2-oxazole-3-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
3-[(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole
(3S,4S)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-methylpiperidine-3,4-diol
5-benzyl-4-(2-methoxyacetyl)-1-(3-phenylphenyl)piperazin-2-one
(2R,6S)-2,6-dimethyl-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)morpholine
(2S,4R)-4-amino-1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
N-{3-[(cyclobutylcarbamoyl)amino]-4-fluorophenyl}propanamide
ethyl 4-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamido]piperidine-1-carboxylate
5-(2,6-difluorophenoxymethyl)-N-[(2,3-dimethoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
2-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridine-3-carboxamide