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4-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}morpholine
4-methyl-6-[4-({[1-(pyrrolidin-1-yl)cyclohexyl]methyl}amino)piperidin-1-yl]pyrimidin-2-amine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3-(1,2-oxazinan-2-yl)propanamide
1-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-2-one
N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(pyridin-2-ylmethyl)-4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
[(3R,4R)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-(propan-2-yl)-4-{2-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1H-pyrazole
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
4-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]-2,1,3-benzoxadiazole
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
N-[2-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)quinolin-5-yl]acetamide
{5-[(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]furan-2-yl}methanol
(3S,4S)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
N-[(3,4-difluorophenyl)methyl]-3-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-3-yl}propanamide
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
N-(1-cyclohexyl-1H-pyrazol-5-yl)-3-(1-methylcyclopropyl)propanamide
4-(1-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,2-diol
3-({1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
4-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]morpholine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-methyl-7-(oxolan-3-ylmethyl)-N-(pyridin-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-(cyclopropylmethyl)-2-[(4-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
(2S,4S)-1-(5-acetylthiophene-2-carbonyl)-4-amino-N-ethylpyrrolidine-2-carboxamide
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-(2-chloro-4-fluoro-5-methylphenyl)-3-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
4-benzoyl-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine
5-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[3-(sulfamoylmethyl)phenyl]propanamide
3-[(3R,4S)-1-(2-methyl-1-benzofuran-7-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N'1-[2-(4-methoxyphenyl)ethyl]-N'1-[(1-methylpiperidin-4-yl)methyl]cyclopropane-1,1-dicarboxamide
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}acetamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-ethyl-N-(2-methylprop-2-en-1-yl)benzamide
14-(quinolin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
5-{1-[2-(3-methylpiperidin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}-2-(thiophen-2-yl)pyrimidine
(3R,4S)-4-cyclopropyl-1-(1-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
N-(dimethyl-1,2-oxazol-4-yl)-2-(trifluoromethyl)morpholine-4-carboxamide
3-chloro-6-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyridazine