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(4aR,8aR)-2-methanesulfonyl-7-[(1-methyl-1H-indol-6-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
4-ethyl-5-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-3-carboxamide
1-{1-[(methylcarbamoyl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
6-hydroxy-N-[2-(3-methylphenoxy)phenyl]-1,4-oxazepane-4-carboxamide
2-(2,5-dichlorophenyl)-6-methylpyridine-3-carboxamide
(2R)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
(2S,4R)-4-amino-1-[(6-acetamidoquinolin-2-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
8-[4-(4-ethylphenyl)butanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{1'-[(2,4-difluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
N-(2-methoxyethyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(4-ethylmorpholin-2-yl)ethyl]-1-benzofuran-2-sulfonamide
1-benzoyl-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
3-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
6-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
5,7-dimethyl-N-[4-(oxolan-2-yl)butyl]pyrido[2,3-d]pyrimidin-4-amine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
(5S)-5-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
[(1-methyl-1H-imidazol-2-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
propyl 4-oxo-2-[(phenylsulfanyl)methyl]-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxylate
2-ethyl-4-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
(4aS,7aR)-N-(3-ethylphenyl)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)[(2,4,5-trimethoxyphenyl)methyl]amine
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]pent-4-enamide
2-[2-(pyridin-2-yl)ethyl]-8-(pyrimidin-5-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1H-indazol-3-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
{1-[(2,4-dimethoxyphenyl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(cyclopropylmethyl)(oxolan-2-ylmethyl)amine
3-(3,5-dimethylphenyl)-N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
1-{1'-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-[cyclohexyl(methyl)amino]-3-[3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)phenoxy]propan-2-ol
5-butyl-1-(2-methoxyphenyl)-4-(1-methyl-1H-pyrazole-5-carbonyl)piperazin-2-one
6-chloro-3-{[3-(hydroxymethyl)piperidin-1-yl]methyl}-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
5-chloro-4,6-dimethyl-3-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
7-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
N-(pyridin-2-ylmethyl)-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
1-[2-(4-fluorophenoxy)acetyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(2-fluorobenzoyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
1-(1-benzylpiperidin-4-yl)-4-[(2-chlorophenyl)methyl]-1,4-diazepan-5-one
1-{5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-methyl-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
N-[2-(benzyloxy)ethyl]-4-methylpyrimidin-2-amine
2-[1-({1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-cyclopropyl-5-(4,4-difluoropiperidine-1-carbonyl)-4-methylpyrimidine
1-(2-ethoxypyridine-3-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-(4-methyl-1,3-thiazole-5-carbonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(3-methylphenyl)acetamide
1-(2H-1,3-benzodioxol-5-yl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
N-[(3-methylpyridin-2-yl)methyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide