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N-{1-azabicyclo[2.2.2]octan-3-yl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
N-(oxolan-2-ylmethyl)-N-propyl-1H-imidazole-2-carboxamide
N-(1-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(2-methylphenoxy)azetidine
2-{5-cyclopropyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2,5-dimethylthiophen-3-yl)pyrimidine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[2-(difluoromethoxy)phenyl]methyl}piperidine
4-chloro-N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-methyl-1H-indole-2-carboxamide
4-[4-(3-methylbenzoyl)piperazin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(3S)-2-oxoazepan-3-yl]-4-(1H-pyrazol-1-yl)-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
3-{2-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclopropylacetamide
2-[(1-cyclopentanecarbonylpiperidin-4-yl)formamido]-N-methyl-2-phenylacetamide
ethyl 3-[(4-fluorophenyl)methyl]-1-(2-hydroxy-6-methylpyridine-3-carbonyl)piperidine-3-carboxylate
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
methyl 2-[methyl({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]acetate
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
7-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methoxy}-2H-chromen-2-one
(1S,5R)-3-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(2-methylpropyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
ethyl 1-(2-hydroxyethyl)-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-({5-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-(3-methoxypropyl)piperidine-3-carboxylic acid
(2R)-2-hydroxy-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
4-(2,4-difluoro-3-methoxyphenyl)-1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-1,2,3-triazole
N-(1-ethyl-1H-pyrazol-5-yl)-2-[4-(4-oxo-3,4-dihydro-2H-1-benzopyran-7-yl)-1H-pyrazol-1-yl]acetamide
5-cyclopropyl-3-[4-(3-methyl-1H-1,2,4-triazol-5-yl)phenyl]-1,2,4-oxadiazole
N-(oxolan-2-ylmethyl)-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)propanamide
5-{3-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
[(2R)-1-(3-chloro-1H-indole-2-carbonyl)pyrrolidin-2-yl]methanol
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N3-cyclohexyl-1-cyclopropyl-N5-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(2,4-dioxoimidazolidin-1-yl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}acetamide
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(3R,4R)-1-(3-chloro-5-methoxybenzoyl)-4-cyclopropyl-3-methylpiperidin-4-ol
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-(3-phenylpropyl)piperidine-4-carboxylate
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-[(3-methoxyphenyl)amino]butanamide
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}acetamide
1-[3-(carbamoylmethoxy)benzoyl]-3-propylpiperidine-3-carboxylic acid
N-methyl-2-(3-methyl-2-oxopyrrolidin-1-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]urea
4-({[(2-chloro-3,6-difluorophenyl)methyl](methyl)amino}methyl)-1-cyclopentylpyrrolidin-2-one
methyl 1-benzyl-3-(furan-3-amido)-5-{[(2-methylphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-(2-methoxyphenyl)piperazin-2-one
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-{5-[(4-methylpiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one