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N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
4-(4-ethyl-1H-pyrazol-5-yl)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
2-cyclopropanecarbonyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-methyl-2-({4-[(1-methylpiperidin-3-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
2-(2,4-dichlorophenoxy)-N-[2-(1H-imidazol-1-yl)propyl]acetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-[2-(pyrrolidin-1-ylmethyl)-4-(thiophen-2-yl)phenoxy]acetamide
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-methylpropan-1-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-2,2-dimethyloxane-4-carboxamide
2-{3-cyclopentyl-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-{1-benzyl-4-[(2-fluoro-5-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 3-[(2-fluorophenyl)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
(1R,7S)-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl 3-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)-5-[(3,3-dimethylbutanamido)methyl]benzoate
2,4-dichloro-6-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}phenol
3-({8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)pyridin-2-amine
[(2-phenoxypyridin-3-yl)methyl](pyridin-4-ylmethyl)amine
1-({1-[5-(ethoxycarbonyl)pyridin-2-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
[(3R,4R)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-amine
2-(4-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
N-ethyl-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidine-3-carboxamide
N-[1-(cyclohexylcarbamoyl)piperidin-4-yl]-2-cyclopropyl-4-hydroxypyrimidine-5-carboxamide
(4S,6R)-N-[4-methoxy-2-(2-methylpropanamido)phenyl]-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
2-{[7-(oxane-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl 3-[7-chloro-2-({pyrazolo[1,5-a]pyrimidin-3-ylformamido}methyl)-2,3-dihydro-1-benzofuran-5-yl]benzoate
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)oxolane-2-carboxamide
4-(4-{[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
4-({4-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-(furan-2-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[2-(thiomorpholine-4-carbonyl)morpholine-4-carbonyl]-1H-indazole
2-{[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]sulfanyl}pyridine
1-(3-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
6-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-cyclopentylpyrimidin-2-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}acetamide
4-methyl-2-propyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-ethoxy-3-{[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propan-2-ol
N-(2-methylpropyl)-3-oxo-N-(thiophen-3-ylmethyl)-3,4-dihydroquinoxaline-2-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-4-(pyrrolidin-1-ylmethyl)-1H-pyrazole
2-methyl-6-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
1-cyclohexyl-4-(3-hydroxy-6-methylpyridin-2-yl)-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
2-acetyl-8-(pyrimidin-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(4-chlorophenyl)-1-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}butan-1-one
N-(2-fluoro-4-methylphenyl)-2-{[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazol-4-yl]formamido}acetamide