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N-[3-(3-methoxyphenyl)phenyl]-1-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxamide
3,5-dihydroxy-4-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylbenzamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-3,4-difluorobenzene-1-sulfonamide
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
5-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-5-oxopentanamide
5-({4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)-2-methoxyphenol
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
N-[2-(3-phenylpiperidin-1-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-(3,4-diethoxybenzoyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-methyl-2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
(1S,6R)-3-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
2-methyl-3-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridine
(4aR,8aR)-1-(2-chloropyridine-4-carbonyl)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridine
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1'-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[(3R,4S)-4-(dimethylamino)-1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl]propan-1-ol
N'1-[(3R,4S)-4-(propan-2-yl)-1-(5-propylpyrimidin-4-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
2-tert-butyl-N-[(2-ethylpyrimidin-5-yl)methyl]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
5-(2-methylpropyl)-1'-[2-(methylsulfanyl)pyrimidin-4-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-benzyl-N3-ethyl-4-oxo-N5-[2-(4-phenylpiperidin-1-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-butyl-N-(6-methoxypyridin-3-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
N-cyclopropyl-2,2-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]oxane-4-carboxamide
2-(4-fluoro-2-methylphenyl)-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)acetamide
7-(2-hydroxyethyl)-2-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(3-methylpyridin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]morpholine
4-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2,3-thiadiazole
4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-3-(1H-imidazol-2-yl)piperidine
N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)-2,3-dihydro-1H-indene-1-carboxamide
4-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
[(3R,4R)-1-(3-chloro-4-methoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-1,2,4-triazole-5-carboxamide
1-benzyl-2-(2-methylpropanesulfonyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
3-(2,5-dioxoimidazolidin-4-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
(1R,9aR)-1-({[2-(3-hydroxy-4-methoxyphenyl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(3S,4S)-1-(2-hydroxybenzoyl)-4-(naphthalen-2-yl)piperidin-3-ol
7-[1-(4-chlorophenyl)cyclohexanecarbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-(2-methoxyquinolin-3-yl)pyridin-3-amine
5-{2-oxo-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
5-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
(2S,4S)-4-amino-1-(cyclopropanesulfonyl)-N-ethylpyrrolidine-2-carboxamide
3-(2-phenylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
2-(2,1,3-benzoxadiazol-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid