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N-[1-(cyclohex-1-en-1-yl)ethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-methyl-2-oxo-5-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridine-3-carbonitrile
2-[(2,6-dichlorophenyl)methyl]-5-(3-propylmorpholine-4-carbonyl)pyrimidin-4-ol
ethyl 4-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]piperidine-1-carboxylate
2-(2,5-dimethylfuran-3-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
5-[1-(2-aminoacetyl)pyrrolidin-2-yl]-N-[3-(methylsulfanyl)phenyl]thiophene-2-carboxamide
2-cyclopropyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrimidine-5-carboxamide
5-chloro-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyridine
2-chloro-5-acetamido-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]benzamide
9-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
2-(dimethylamino)-7-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-methoxy-2-methyl-5-[6-(piperidine-1-carbonyl)pyrazin-2-yl]quinoline
(1R,5R)-N,N-dimethyl-6-(2-phenoxyacetyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-[4-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
4-[(2-chlorophenyl)methyl]-1-(3-methylpyrazin-2-yl)piperidine-4-carboxylic acid
4-({2-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}acetamide
3-hydroxy-1-(2-methoxyethyl)-3-({[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
5-{5-[1-(furan-2-ylmethyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
3-[(oxolan-2-ylmethyl)(2-phenoxyethyl)carbamoyl]benzoic acid
1-[(2E)-2-methylbut-2-enoyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
({4-cyclopropyl-5-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-(4-methanesulfonylpiperazine-1-carbonyl)-N-phenylpyrimidin-2-amine
N-[(2-{3-[2-(4-methoxyphenyl)acetamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
N-{1-[({[1-(morpholin-4-yl)cyclopentyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}furan-2-carboxamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(thiophen-3-yl)acetyl]piperidine-4-carboxylic acid
9-(2-methyl-6-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(furan-3-ylmethyl)amino]-5-(phenylsulfamoyl)-N-(pyridin-3-ylmethyl)benzamide
N-methyl-1-(2-methyl-6-propylpyrimidin-4-yl)-N-(oxan-2-ylmethyl)piperidin-4-amine
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(furan-2-carbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-(piperidin-4-yl)pyrimidin-2-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-hydroxyethyl)-N-propylacetamide
2-fluoro-N-(1,2-oxazol-3-ylmethyl)-5-sulfamoylbenzamide
2-[4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]ethan-1-ol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-{2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}acetamide
1-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
2-cyclopropyl-9-(2,6-difluoro-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
3-[2-(methylsulfanyl)phenyl]-[1,2,4]triazolo[4,3-a]pyridine
3-{[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}benzonitrile
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-benzyl-1-{1,9-dioxaspiro[5.5]undecan-4-yl}piperidine-4-carboxamide
(1S,5R)-3-(oxan-4-yl)-6-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane