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4-chloro-2-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)phenol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-1-benzoxepine-4-carboxamide
1-{1-[5-(2-methylphenyl)-1,2,4-triazin-3-yl]-4-phenylpiperidin-4-yl}ethan-1-one
3-(pentan-2-yl)-8-(quinoline-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-[(4-methylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(2-hydroxypropyl)benzamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
N-cyclopropyl-2-methyl-N-(1,3-thiazol-5-ylmethyl)-1,3-thiazole-4-carboxamide
2-(3-methoxypiperidin-1-yl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
4-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-cyclooctyl-4-oxobutanamide
2-fluoro-6-methoxy-N-(3-methoxy-2,2-dimethylpropyl)benzamide
N-[2-(1H-indol-3-yl)ethyl]-2-(2-methylbenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
(2S)-2-[4-(3,4-dimethoxyphenyl)-1H-1,2,3-triazol-1-yl]-4-methylpentan-1-ol
4-(5-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-methyl-N-(oxan-2-ylmethyl)-9-oxo-9,10-dihydroacridine-4-carboxamide
ethyl 2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}pyridine-3-carboxylate
2-[(3,5-difluorophenyl)methyl]-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
2-[(4-ethoxy-3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-(2-methoxyphenyl)-1-[2-(pent-4-enamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridine-2,4-diol
2-[2-(1H-imidazol-4-yl)ethyl]-9-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
N2,N2-dimethyl-N4-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(4-fluorophenyl)methyl]-3-methoxy-N-methylbenzamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
1-(2-methylphenyl)-3-[1-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
7-(1-phenylcyclopentanecarbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3aS,6aR)-5-(dimethyl-1,3-thiazole-5-carbonyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-methyl-N-[4-(morpholin-4-yl)butyl]-4-(pyridin-3-yl)pyrimidin-2-amine
6-chloro-2-{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carboxamide
(1S,5R)-3-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3-thiazol-2-amine
(3R,5S)-1-benzyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(2-phenylethyl)piperidine-3-carboxamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
N-[(6-methylpyridin-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-(2-chlorophenyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-one
N-[1-(3-chlorophenyl)cyclopropyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(2-ethoxypyridin-3-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-benzyl-3-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyrrolidine-2-carboxamide
N-benzyl-2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]acetamide
N-{1-[3-methyl-1-(naphthalen-2-yl)-1H-1,2,4-triazol-5-yl]propan-2-yl}acetamide
1-{1'-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one