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[(3R,4R)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-(4-{[(5-chlorothiophen-2-yl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-butyl-6-methyl-2-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydropyridine-3-carboxamide
3-(4-chlorobenzoyl)-1-(1,4-dithiepan-6-yl)piperidine
N-cyclopentyl-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)thiophene-2-carboxamide
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3-carboxamide
4-acetamido-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-[(5-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}thiophen-2-yl)formamido]acetamide
(1S,5R)-6-(5-chloro-2-methylbenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
(4aS,7aR)-1-[(2-methoxyphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)morpholine-2-carboxamide
N-ethyl-N-methyl-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-(4-{[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
methyl 2-(cyclopentylamino)-2-(3-methylphenyl)acetate
2-phenoxy-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
6-(morpholin-4-yl)-N-[2-(pyridin-3-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-phenyl-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperazine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(thian-4-yl)piperazin-1-yl]ethan-1-one
2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrazine
2-{4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
(3S,4S)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][2-(7-methyl-1H-indol-3-yl)ethyl]amine
7-(cyclopropylmethyl)-N-[4-(methylsulfanyl)phenyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-[2-(4-fluorophenyl)piperidine-1-carbonyl]pyridin-4-amine
1'-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]phenoxy}pyridine
4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1-phenylbutan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(3-fluorophenyl)methyl]piperidin-4-ol
1-{3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propyl}-1H-1,2,3,4-tetrazole
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1-methyl-1H-indole
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
5-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-{[1-(pyridin-2-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-{[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(3R,9aR)-3-(propan-2-yl)-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
3-{2-[(2-methyl-1,3-thiazol-5-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
4-acetyl-N-[3-(3-methoxyphenyl)phenyl]-1,4-diazepane-1-carboxamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-ol
2-[7-(2-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]-N-(4-methylphenyl)acetamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}pyrrolidin-3-amine
2-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
1-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine